SCHEMBL9684571

SCHEMBL9684571

CCOC(=O)c1cnc(N2CCNCC2)nc1C(=O)OCC

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.49
DYRK1A Q13627 1/20 0.48
MAPT P10636 2/20 0.47
POLB P06746 2/20 0.47
ALDH1A1 P00352 2/20 0.47
MEN1 O00255 2/20 0.46
KMT2A Q03164 2/20 0.46
KDM4E B2RXH2 2/20 0.46
ALOX15 P16050 1/20 0.44
HSP90AA1 P07900 1/20 0.44
HSP90AB1 P08238 1/20 0.44
PDE4B Q07343 1/20 0.44
TSHR P16473 2/20 0.44
GAA P10253 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
HPGD P15428 1/20 0.43
CASP1 P29466 1/20 0.43
CYP2C19 P33261 1/20 0.43
CASP7 P55210 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21477192 0.87 MEN1 (0.53) MAPTPOLBALDH1A1MEN1KMT2A
SCHEMBL12929334 0.85 ALDH1A1 (0.59) ADORA3DYRK1AMAPTPOLBALDH1A1
SCHEMBL11822825 0.83 MEN1 (0.51) ADORA3DYRK1AMAPTPOLBALDH1A1
SCHEMBL11822073 0.83 MEN1 (0.51) ADORA3DYRK1AMAPTPOLBALDH1A1
SCHEMBL11824584 0.83 ALOX15 (0.67) ADORA3MAPTPOLBALDH1A1MEN1
SCHEMBL11825216 0.82 MEN1 (0.50) ADORA3DYRK1AMAPTPOLBALDH1A1
SCHEMBL11825199 0.82 MEN1 (0.50) ADORA3DYRK1AMAPTPOLBALDH1A1
SCHEMBL11873704 0.82 ADORA3 (0.44) ADORA3DYRK1AMAPTPOLBALDH1A1
SCHEMBL386644 0.81 OGA (0.50) ADORA3DYRK1AMAPTPOLBALDH1A1
SCHEMBL11819432 0.81 MEN1 (0.49) ADORA3DYRK1AMAPTPOLBALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188094-B1 QUINAZOLINE DERIVATIVES AND ANTIHYPERTENSIVE PREPARATIONS CONTAINING SAME AS EFFECTIVE COMPONENTS MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1992-03-18 EP disclosed
US-4734418-A Quinazoline compounds and antihypertensives MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1988-03-29 US disclosed
EP-0188094-A2 Quinazoline derivatives and antihypertensive preparations containing same as effective components MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1986-07-23 EP disclosed