SCHEMBL9685239

SCHEMBL9685239

CCNC(=O)c1cnc(N2CCN(Cc3ccccc3)CC2)nc1C

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.60
PTPN11 Q06124 2/20 0.51
HDAC6 Q9UBN7 2/20 0.48
MAPT P10636 2/20 0.48
LMNA P02545 2/20 0.47
HTT P42858 2/20 0.47
ALDH1A1 P00352 2/20 0.47
KDM4E B2RXH2 1/20 0.47
CHRM4 P08173 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
POLB P06746 1/20 0.46
HDAC3 O15379 1/20 0.46
HDAC4 P56524 1/20 0.46
HDAC1 Q13547 1/20 0.46
HDAC7 Q8WUI4 1/20 0.46
HDAC2 Q92769 1/20 0.46
HDAC10 Q969S8 1/20 0.46
HDAC11 Q96DB2 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9686641 0.90 TRPA1 (0.57) TRPA1PTPN11HDAC6MAPTLMNA
SCHEMBL9685113 0.90 TRPA1 (0.58) TRPA1PTPN11HDAC6LMNAHTT
SCHEMBL9685390 0.89 TRPA1 (0.60) TRPA1PTPN11HDAC6LMNAHTT
SCHEMBL9685139 0.87 TRPA1 (0.56) TRPA1PTPN11LMNAHTTALDH1A1
SCHEMBL9684387 0.85 TRPA1 (0.55) TRPA1PTPN11MAPTLMNAHTT
SCHEMBL9686160 0.84 TRPA1 (0.54) TRPA1PTPN11LMNAHTTALDH1A1
SCHEMBL9686157 0.84 NPSR1 (0.55) TRPA1PTPN11MAPTLMNAHTT
SCHEMBL9686804 0.83 TRPA1 (0.52) TRPA1LMNAHTTALDH1A1SMN1; SMN2
SCHEMBL9685068 0.80 TRPA1 (0.64) TRPA1PTPN11HDAC6MAPTLMNA
SCHEMBL9685091 0.78 TRPA1 (0.59) TRPA1PTPN11MAPTLMNAHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0188094-B1 QUINAZOLINE DERIVATIVES AND ANTIHYPERTENSIVE PREPARATIONS CONTAINING SAME AS EFFECTIVE COMPONENTS MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1992-03-18 EP disclosed
US-4734418-A Quinazoline compounds and antihypertensives MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1988-03-29 US disclosed
EP-0188094-A2 Quinazoline derivatives and antihypertensive preparations containing same as effective components MITSUI PETROCHEMICAL INDUSTRIES, LTD. (JP) 1986-07-23 EP disclosed