SCHEMBL9685844

SCHEMBL9685844

CN(O)C(=O)NCCc1cc2ccccc2o1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 2/20 0.46
HSD17B10 Q99714 2/20 0.46
NPC1 O15118 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
ESR1 P03372 1/20 0.43
ESR2 Q92731 1/20 0.43
NAMPT P43490 1/20 0.43
LOXL2 Q9Y4K0 1/20 0.43
ACKR3 P25106 1/20 0.43
OPRM1 P35372 1/20 0.43
OPRK1 P41145 1/20 0.43
TMEM97 Q5BJF2 1/20 0.43
SIGMAR1 Q99720 1/20 0.43
MEN1 O00255 2/20 0.43
KMT2A Q03164 2/20 0.43
RAB9A P51151 1/20 0.43
HPGD P15428 2/20 0.42
SMN1; SMN2 Q16637 3/20 0.41
TP53 P04637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4499441 0.83 MTNR1A (0.53) ALDH1A1KDM4EHSD17B10NPC1L3MBTL1
SCHEMBL9684718 0.79 NPC1 (0.47) ALDH1A1HSD17B10NPC1L3MBTL1ESR1
SCHEMBL7568119 0.75 HDAC1 (0.41) ALDH1A1HSD17B10NPC1L3MBTL1ESR1
SCHEMBL10662358 0.75 LOXL2 (0.55) L3MBTL1LOXL2SMN1; SMN2MAOB
SCHEMBL31173757 0.75 LOXL2 (0.55) L3MBTL1LOXL2SMN1; SMN2MAOB
SCHEMBL2396386 0.73 LOXL2 (0.46) ALDH1A1KDM4EHSD17B10L3MBTL1ESR1
SCHEMBL9666803 0.73 CES2 (0.53) ALDH1A1KDM4EHSD17B10OPRM1SIGMAR1
SCHEMBL30886917 0.71 SMN1; SMN2 (0.57) ALDH1A1KDM4EHSD17B10L3MBTL1LOXL2
SCHEMBL10368235 0.71 LOXL2 (0.55) KDM4ENPC1ESR1ESR2LOXL2
SCHEMBL15980824 0.71 CYP2D6 (0.58) NPC1L3MBTL1LOXL2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1990008545-A1 LIPOXYGENASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1990-08-09 WO claimed
US-5175183-A Antiinflammatory agents, respiratory system disorders ABBOTT LABORATORIES (US) 1992-12-29 US disclosed
WO-1990008545-A1 LIPOXYGENASE INHIBITING COMPOUNDS ABBOTT LABORATORIES (US) 1990-08-09 WO disclosed