SCHEMBL9686613

SCHEMBL9686613

CC1=C(C)C(=O)N(c2ccc3c(c2)N(Cc2ccon2)C(=O)CO3)C1=O

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.43
HTT P42858 2/20 0.41
TSHR P16473 1/20 0.41
PLK1 P53350 1/20 0.39
PIK3CG P48736 3/20 0.38
ALDH1A1 P00352 2/20 0.38
USP2 O75604 1/20 0.38
ALOX15 P16050 1/20 0.38
CYP1B1 Q16678 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
CYP2C19 P33261 1/20 0.36
GAA P10253 1/20 0.36
SLC5A1 P13866 2/20 0.36
SLC5A2 P31639 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9687032 0.87 BRD4 (0.36) BRD4HTTTSHRPIK3CGCYP1B1
SCHEMBL9686626 0.81 HDAC4 (0.41) BRD4HTTTSHRPLK1PIK3CG
SCHEMBL9832981 0.79 HTT (0.49) BRD4HTTTSHRPLK1PIK3CG
SCHEMBL9831606 0.77 PLK1 (0.45) BRD4HTTTSHRPLK1PIK3CG
SCHEMBL9831062 0.77 HTT (0.44) BRD4HTTTSHRPLK1ALDH1A1
SCHEMBL9872261 0.73 NMT1 (0.37) BRD4HTTTSHRPIK3CGALDH1A1
SCHEMBL9686487 0.73 CYP1B1 (0.36) CYP1B1
SCHEMBL9687722 0.72 HDAC4 (0.39) BRD4HTTTSHRPLK1PIK3CG
SCHEMBL9687661 0.71 BRD4 (0.54) BRD4TSHRPIK3CGALDH1A1ALOX15
SCHEMBL9687801 0.67 BRD4 (0.57) BRD4TSHRALDH1A1ALOX15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0296416-B1 BENZO-ANELLATED CYCLIC COMPOUNDS NIHON BAYER AGROCHEM K.K. (JP) 1992-07-29 EP disclosed
US-5077401-A Herbicides NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1991-12-31 US disclosed
US-4902335-A Benzo-fused cyclic compounds NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1990-02-20 US disclosed
EP-0296416-A1 Benzo-anellated cyclic compounds NIHON BAYER AGROCHEM K.K. (JP) 1988-12-28 EP disclosed