SCHEMBL9687722

SCHEMBL9687722

Cc1nc(CN2C(=O)COc3ccc(N4C(=O)C5=C(CCCC5)C4=O)cc32)no1

nearest known ligand 0.60

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
TSHR P16473 1/20 0.38
HTT P42858 1/20 0.38
PIK3CG P48736 2/20 0.37
PLK1 P53350 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
SLC5A1 P13866 3/20 0.35
SLC5A2 P31639 3/20 0.35
BRD4 O60885 2/20 0.35
GRM5 P41594 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9686626 0.90 HDAC4 (0.41) HDAC4HDAC1HDAC6TSHRHTT
SCHEMBL9687032 0.80 BRD4 (0.36) TSHRHTTPIK3CGSLC5A1SLC5A2
SCHEMBL9687661 0.77 BRD4 (0.54) HDAC1HDAC6TSHRPIK3CGBRD4
SCHEMBL4075188 0.75 TSHR (0.38) TSHRHTTPLK1CYP1A2CYP3A4
SCHEMBL9686469 0.73 NMT1 (0.41) HDAC4HDAC1HDAC6TSHRHTT
SCHEMBL9423272 0.72 SLC5A1 (0.38) TSHRHTTPLK1CYP3A4CYP2D6
SCHEMBL9686613 0.72 BRD4 (0.43) TSHRHTTPIK3CGPLK1CYP1A2
SCHEMBL9685814 0.70 TERT (0.44) HDAC4HDAC1HDAC6TSHRSLC5A1
SCHEMBL9832981 0.68 HTT (0.49) TSHRHTTPIK3CGPLK1SLC5A1
SCHEMBL9686487 0.67 CYP1B1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0296416-B1 BENZO-ANELLATED CYCLIC COMPOUNDS NIHON BAYER AGROCHEM K.K. (JP) 1992-07-29 EP disclosed
US-5077401-A Herbicides NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1991-12-31 US disclosed
US-4902335-A Benzo-fused cyclic compounds NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1990-02-20 US disclosed
EP-0296416-A1 Benzo-anellated cyclic compounds NIHON BAYER AGROCHEM K.K. (JP) 1988-12-28 EP disclosed