SCHEMBL9686626

SCHEMBL9686626

CC1=C(C)C(=O)N(c2ccc3c(c2)N(Cc2noc(C)n2)C(=O)CO3)C1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC6 Q9UBN7 1/20 0.41
HTT P42858 2/20 0.40
TSHR P16473 1/20 0.40
BRD4 O60885 2/20 0.39
PLK1 P53350 1/20 0.38
PIK3CG P48736 3/20 0.37
GRM5 P41594 1/20 0.37
USP2 O75604 1/20 0.36
ALDH1A1 P00352 1/20 0.36
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C19 P33261 1/20 0.35
GAA P10253 1/20 0.35
SLC5A1 P13866 2/20 0.35
SLC5A2 P31639 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9687722 0.90 HDAC4 (0.39) HDAC4HDAC1HDAC6HTTTSHR
SCHEMBL9686613 0.81 BRD4 (0.43) HTTTSHRBRD4PLK1PIK3CG
SCHEMBL9832981 0.78 HTT (0.49) HTTTSHRBRD4PLK1PIK3CG
SCHEMBL9686469 0.76 NMT1 (0.41) HDAC4HDAC1HDAC6HTTTSHR
SCHEMBL9831606 0.76 PLK1 (0.45) HTTTSHRBRD4PLK1PIK3CG
SCHEMBL9831062 0.76 HTT (0.44) HTTTSHRBRD4PLK1USP2
SCHEMBL9685814 0.73 TERT (0.44) HDAC4HDAC1HDAC6TSHRBRD4
SCHEMBL9687032 0.69 BRD4 (0.36) HTTTSHRBRD4PIK3CGSLC5A1
SCHEMBL9687661 0.65 BRD4 (0.54) HDAC1HDAC6TSHRBRD4PIK3CG
SCHEMBL24258037 0.65 HDAC1 (0.61) HDAC4HDAC1HDAC6TSHRGRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0296416-B1 BENZO-ANELLATED CYCLIC COMPOUNDS NIHON BAYER AGROCHEM K.K. (JP) 1992-07-29 EP disclosed
US-5077401-A Herbicides NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1991-12-31 US disclosed
US-4902335-A Benzo-fused cyclic compounds NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1990-02-20 US disclosed