SCHEMBL9687032

SCHEMBL9687032

O=C1COc2ccc(N3C(=O)C4=C(CCCC4)C3=O)cc2N1Cc1ccon1

nearest known ligand 0.64

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.36
SLC5A1 P13866 4/20 0.36
SLC5A2 P31639 4/20 0.36
PIK3CG P48736 4/20 0.36
TSHR P16473 1/20 0.35
HTT P42858 1/20 0.35
CYP1B1 Q16678 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
KMO O15229 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9686613 0.87 BRD4 (0.43) BRD4SLC5A1SLC5A2PIK3CGTSHR
SCHEMBL9686487 0.86 CYP1B1 (0.36) CYP1B1
SCHEMBL9687661 0.84 BRD4 (0.54) BRD4PIK3CGTSHRL3MBTL1
SCHEMBL9687722 0.80 HDAC4 (0.39) BRD4SLC5A1SLC5A2PIK3CGTSHR
SCHEMBL4075188 0.78 TSHR (0.38) TSHRHTTKMO
SCHEMBL9423272 0.75 SLC5A1 (0.38) BRD4SLC5A1SLC5A2TSHRHTT
SCHEMBL9872261 0.72 NMT1 (0.37) BRD4PIK3CGTSHRHTTCYP1B1
SCHEMBL9686626 0.69 HDAC4 (0.41) BRD4SLC5A1SLC5A2PIK3CGTSHR
SCHEMBL9685904 0.69 BRD4 (0.49) BRD4TSHR
SCHEMBL9687072 0.67 CYP1B1 (0.35) BRD4CYP1B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0296416-B1 BENZO-ANELLATED CYCLIC COMPOUNDS NIHON BAYER AGROCHEM K.K. (JP) 1992-07-29 EP disclosed
US-5077401-A Herbicides NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1991-12-31 US disclosed
US-4902335-A Benzo-fused cyclic compounds NIHON TOKUSHU NOYAKU SEIZO K.K. (JP) 1990-02-20 US disclosed
EP-0296416-A1 Benzo-anellated cyclic compounds NIHON BAYER AGROCHEM K.K. (JP) 1988-12-28 EP disclosed