SCHEMBL9687013

SCHEMBL9687013

CCc1c(C=O)cc(C(=O)[O-])c(O)c1OC.CCc1c(C=O)cc(C(=O)[O-])c(O)c1OC.[Ca+2]

nearest known ligand 0.38

Known targets — ChEMBL curated mechanism

GABBR1GABBR2GABRA1GABRA2GABRA3GABRA4GABRA5GABRA6GABRB1GABRB2GABRB3GABRDGABREGABRG1GABRG2GABRG3GABRPGABRQGRIN1GRIN2AGRIN2BGRIN2CGRIN2DGRIN3AGRIN3BHMGCRMMP1MMP13MMP7MMP8PTGS1PTGS2ileSpolrplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of None. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 14/20 0.38
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
ALDH1A1 P00352 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C19 P33261 1/20 0.34
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.33
MCL1 Q07820 1/20 0.33
TRIM24 O15164 1/20 0.33
TYR P14679 1/20 0.33
TRIM33 Q9UPN9 1/20 0.33
TLR2 O60603 1/20 0.33
TLR1 Q15399 1/20 0.33
TLR6 Q9Y2C9 1/20 0.33
TDP1 Q9NUW8 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Potassium Ion SCHEMBL9686356 0.97 ERN1 (0.38) ERN1CA1CA2ALDH1A1CYP1A2
SCHEMBL9688193 0.97 ERN1 (0.38) ERN1CA1CA2ALDH1A1CYP1A2
SCHEMBL9687459 0.97 ERN1 (0.38) ERN1CA1CA2ALDH1A1CYP1A2
SCHEMBL4755047 0.86 MAPT (0.43) ERN1CA1CA2MAPTLMNA
SCHEMBL1940680 0.79 ERN1 (0.44) ERN1CA1CA2MAPTLMNA
SCHEMBL14542987 0.76 ERN1 (0.37) ERN1CA1CA2MAPTLMNA
SCHEMBL4757842 0.73 MAPT (0.42) ERN1CA1CA2MAPTLMNA
SCHEMBL4755033 0.72 MAPT (0.41) ERN1CA1CA2MAPTLMNA
SCHEMBL29818618 0.69 ALDH1A1 (0.37) ERN1CA1CA2ALDH1A1CYP1A2
SCHEMBL1396832 0.68 CA1 (0.54) ERN1CA1CA2ALDH1A1TRIM24

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0514202-A2 Smoking compositions containing a vanillin-release additive Philip Morris Products Inc. (US) 1992-11-19 EP claimed
US-5144965-A Vanillin carboxylate type additive pyrolyzes to ethyl vanillin; cigarettes PHILIP MORRIS INCORPORATED (US) 1992-09-08 US claimed
EP-0514202-A2 Smoking compositions containing a vanillin-release additive Philip Morris Products Inc. (US) 1992-11-19 EP disclosed
US-5144965-A Vanillin carboxylate type additive pyrolyzes to ethyl vanillin; cigarettes PHILIP MORRIS INCORPORATED (US) 1992-09-08 US disclosed