SCHEMBL9687803

SCHEMBL9687803

COc1cc(N)c([N+](=O)[O-])c(OC(F)F)c1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.47
HTT P42858 2/20 0.42
TDP1 Q9NUW8 4/20 0.41
MCL1 Q07820 1/20 0.39
GRIN2D O15399 1/20 0.37
GRIN3B O60391 1/20 0.37
GRIN1 Q05586 1/20 0.37
GRIN2A Q12879 1/20 0.37
GRIN2B Q13224 1/20 0.37
GRIN2C Q14957 1/20 0.37
GRIN3A Q8TCU5 1/20 0.37
POLB P06746 3/20 0.37
KDM4E B2RXH2 3/20 0.37
CTDSP1 Q9GZU7 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
PTGS2 P35354 1/20 0.37
TUBB4A P04350 1/20 0.35
TUBB P07437 1/20 0.35
TUBA3C P0DPH7 1/20 0.35
TUBA1B P68363 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2905398 0.86 PKM (0.59) PKMHTTTDP1MCL1GRIN2D
SCHEMBL9687963 0.77 PKM (0.47) PKMHTTPOLBALDH1A1LMNA
Hydrochloric Acid SCHEMBL9688513 0.75 POLB (0.39) POLBKDM4ETUBB4ATUBBTUBA3C
SCHEMBL9531415 0.74 ALDH1A1 (0.46) HTTTDP1POLBKDM4EL3MBTL1
SCHEMBL9687879 0.73 PTGS2 (0.50) PKMHTTTDP1PTGS2TUBB4A
SCHEMBL9348700 0.71 PKM (0.65) PKMHTTTDP1MCL1GRIN2D
SCHEMBL622685 0.70 TDP1 (0.57) PKMHTTTDP1MCL1POLB
SCHEMBL16052765 0.70 HTT (0.50) PKMHTTTDP1MCL1GRIN2D
SCHEMBL18246981 0.69 TDP1 (0.49) HTTTDP1POLBKDM4ECTDSP1
SCHEMBL16689316 0.68 ALDH1A1 (0.54) PKMHTTTDP1MCL1GRIN2D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0201575-B1 NEW PICOLINE DERIVATIVES, PREPARATION PROCESS THEREOF, UTILIZATION THEREOF AND DRUGS CONTAINING THEM Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1992-08-12 EP disclosed
US-4686230-A Picoline derivative useful as gastric acid secretion inhibitors BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1987-08-11 US disclosed
US-4675397-A MICROBIOCIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1987-06-23 US disclosed
US-4665067-A BACTERICIDES TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1987-05-12 US disclosed