SCHEMBL9687963

SCHEMBL9687963

COc1cc(NC(C)=O)c([N+](=O)[O-])c(OC(F)F)c1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 3/20 0.47
LMNA P02545 3/20 0.39
ALDH1A1 P00352 2/20 0.39
ABCB1 P08183 3/20 0.38
ABCC1 P33527 3/20 0.38
HTT P42858 2/20 0.38
EPHX1 P07099 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
POLB P06746 2/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
GALR2 O43603 1/20 0.38
MITF O75030 1/20 0.38
HSP90AA1 P07900 1/20 0.38
HPGD P15428 1/20 0.38
XBP1 P17861 1/20 0.38
CCR6 P51684 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ATM Q13315 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10510922 0.81 PKM (0.49) PKMLMNAALDH1A1ABCB1ABCC1
SCHEMBL9528380 0.78 LMNA (0.44) LMNAALDH1A1HTTKMT2APOLB
SCHEMBL9687803 0.77 PKM (0.47) PKMLMNAALDH1A1HTTPOLB
SCHEMBL10668450 0.76 KMT2A (0.41) PKMLMNAALDH1A1HTTKMT2A
SCHEMBL9527341 0.74 LMNA (0.48) PKMLMNAALDH1A1HTTKMT2A
SCHEMBL28878765 0.73 GRIN2D (0.45) PKMLMNAALDH1A1ABCB1ABCC1
SCHEMBL2902495 0.72 ALDH1A1 (0.54) PKMLMNAALDH1A1HTTKMT2A
SCHEMBL7953766 0.72 KMT2A (0.53) PKMLMNAALDH1A1HTTEPHX1
SCHEMBL2848578 0.72 ALDH1A1 (0.47) PKMLMNAALDH1A1HTTEPHX1
SCHEMBL31423349 0.70 ALDH1A1 (0.56) PKMLMNAALDH1A1HTTEPHX1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0201575-B1 NEW PICOLINE DERIVATIVES, PREPARATION PROCESS THEREOF, UTILIZATION THEREOF AND DRUGS CONTAINING THEM Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1992-08-12 EP disclosed
US-4686230-A Picoline derivative useful as gastric acid secretion inhibitors BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1987-08-11 US disclosed