SCHEMBL9688201

SCHEMBL9688201

Clc1ncc(-c2ccccn2)c(-c2ccccn2)n1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR1 P32246 3/20 0.46
CCR5 P51681 3/20 0.46
CCR8 P51685 3/20 0.46
KDM4E B2RXH2 8/20 0.45
LMNA P02545 3/20 0.45
METAP1 P53582 2/20 0.45
CYP1A2 P05177 2/20 0.45
POLB P06746 1/20 0.45
BLM P54132 1/20 0.45
HIF1A Q16665 1/20 0.45
DOHH Q9BU89 1/20 0.45
P4HTM Q9NXG6 1/20 0.45
TP53 P04637 5/20 0.44
SMN1; SMN2 Q16637 4/20 0.44
L3MBTL1 Q9Y468 3/20 0.44
TDP1 Q9NUW8 2/20 0.44
ALOX15 P16050 2/20 0.44
HTT P42858 2/20 0.44
ALPL P05186 1/20 0.44
HSP90AA1 P07900 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5912535 0.84 CCR1 (0.47) CCR1CCR5CCR8KDM4ELMNA
SCHEMBL4540085 0.81 KDM4E (0.54) CCR1CCR5CCR8KDM4ELMNA
SCHEMBL6824538 0.79 KDM4E (0.50) CCR1CCR5CCR8KDM4ELMNA
SCHEMBL8518595 0.76 DHODH (0.45) CCR1CCR5CCR8KDM4ELMNA
SCHEMBL21313138 0.75 KDM4E (0.44) CCR1CCR5CCR8KDM4ELMNA
SCHEMBL5595484 0.72 KDM4E (0.50) CCR1CCR5CCR8KDM4ELMNA
SCHEMBL323086 0.71 KDM4E (0.68) CCR1CCR5CCR8KDM4ELMNA
SCHEMBL31439134 0.71 KDM4E (0.54) CCR1CCR5CCR8KDM4ELMNA
SCHEMBL1513860 0.71 KDM4E (0.54) CCR1CCR5CCR8KDM4ELMNA
SCHEMBL2507724 0.71 KDM4E (0.54) CCR1CCR5CCR8KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120843-A Nervous system disorders UPJOHN (US) 1992-06-09 US disclosed
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP disclosed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP disclosed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO disclosed