SCHEMBL9688433

SCHEMBL9688433

CCOC(=O)Oc1ccc(Br)o1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
POLB P06746 4/20 0.48
KDM4E B2RXH2 4/20 0.48
NPSR1 Q6W5P4 1/20 0.48
GPR55 Q9Y2T6 1/20 0.48
ALDH1A1 P00352 7/20 0.43
PKM P14618 1/20 0.43
CUL4A Q13619 1/20 0.42
KMT2A Q03164 7/20 0.41
MEN1 O00255 3/20 0.41
TSHR P16473 4/20 0.40
MAPK1 P28482 3/20 0.39
LMNA P02545 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2C19 P33261 1/20 0.39
MAPT P10636 4/20 0.39
HPGD P15428 4/20 0.39
SMN1; SMN2 Q16637 2/20 0.39
HSD17B10 Q99714 2/20 0.39
ALOX15 P16050 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7253599 0.80 KMT2A (0.44) POLBKDM4EALDH1A1PKMCUL4A
SCHEMBL9575010 0.80 KMT2A (0.39) POLBKDM4ENPSR1GPR55ALDH1A1
SCHEMBL2486696 0.75 CUL4A (0.47) POLBKDM4ENPSR1GPR55ALDH1A1
SCHEMBL362159 0.71 TSHR (0.63) POLBKDM4ENPSR1GPR55ALDH1A1
SCHEMBL2484716 0.71 CUL4A (0.41) KDM4ENPSR1ALDH1A1CUL4AKMT2A
SCHEMBL2323034 0.71 ALDH1A1 (0.50) POLBGPR55ALDH1A1CUL4AKMT2A
SCHEMBL10973674 0.70 MMP1 (0.44) POLBKDM4EALDH1A1PKMKMT2A
SCHEMBL24418978 0.69 KMT2A (0.49) POLBNPSR1ALDH1A1KMT2AMEN1
SCHEMBL363895 0.69 ALDH1A1 (0.40) POLBALDH1A1PKMCUL4AKMT2A
SCHEMBL4435828 0.69 KDM4E (0.44) POLBKDM4ENPSR1GPR55ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016184652-A9 METHODS FOR PRODUCING METALATED ORGANIC COMPOUNDS LUDWIG-MAXIMILIANS-UNIVERSITÄT MÜNCHEN (DE) 2017-08-10 WO disclosed
EP-0237467-B1 HETEROARYL-OXY-BETA-CARBOLINE DERIVATIVES, THEIR PREPARATION AND USE AS MEDICAMENTS SCHERING AKTIENGESELLSCHAFT (DE) 1992-10-28 EP disclosed
EP-0237467-A2 Heteroaryl-oxy-beta-carboline derivatives, their preparation and use as medicaments SCHERING AKTIENGESELLSCHAFT (DE) 1987-09-16 EP disclosed