SCHEMBL9688536

SCHEMBL9688536

COc1cc(CCN)cc2c(O)n[nH]c12

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 3/20 0.49
TSHR P16473 2/20 0.49
MAPK1 P28482 1/20 0.49
HTR2A P28223 4/20 0.49
HTR2C P28335 2/20 0.49
HTR2B P41595 2/20 0.49
LMNA P02545 2/20 0.48
GLA P06280 1/20 0.48
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
NFKB1 P19838 1/20 0.44
KDM4E B2RXH2 1/20 0.44
ATM Q13315 1/20 0.44
MEN1 O00255 1/20 0.43
APEX1 P27695 1/20 0.43
KMT2A Q03164 1/20 0.43
PTPN1 P18031 1/20 0.37
CYP19A1 P11511 1/20 0.35
TNKS2 Q9H2K2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9688873 0.80 TAAR1 (0.42) TAAR1TSHRMAPK1LMNAGLA
SCHEMBL9688860 0.80 SIGMAR1 (0.41) TSHRHTR2AHTR2BCYP3A4NFKB1
SCHEMBL9687908 0.76 MTNR1A (0.42) TSHRMAPK1
SCHEMBL1467120 0.72 HTR2A (0.68) TAAR1TSHRMAPK1HTR2AHTR2C
Hydrochloric Acid SCHEMBL7370392 0.71 TAAR1 (0.68) TAAR1TSHRMAPK1HTR2AHTR2C
SCHEMBL10041296 0.71 TSHR (0.70) TAAR1TSHRMAPK1HTR2AHTR2C
SCHEMBL9689788 0.71 HTR2A (0.51) TAAR1TSHRMAPK1HTR2AHTR2C
SCHEMBL31079463 0.69 HTR2A (0.68) TAAR1TSHRMAPK1HTR2AHTR2C
SCHEMBL9689779 0.69 HTR2A (0.43) TAAR1TSHRMAPK1HTR2ALMNA
SCHEMBL25374970 0.67 HTR2A (0.76) TAAR1TSHRMAPK1HTR2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0189473-B1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1992-05-27 EP disclosed
US-4958026-A HYPOTENSIVE AGENTS SCHERING AKTIENGESLLSCHAFT (DE) 1990-09-18 US disclosed
EP-0189473-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS. SCHERING AG (DE) 1986-08-06 EP disclosed
WO-1986001204-A1 NEW DOPAMINE DERIVATIVES, PROCESS FOR THEIR PRODUCTION, AND THEIR USE AS MEDICINAL PRODUCTS SCHERING AKTIENGESELLSCHAFT (DE) 1986-02-27 WO disclosed