SCHEMBL9688625

SCHEMBL9688625

Nc1nc(N)c(CCCNc2ccc(C(=O)O)cc2)c(=O)[nH]1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
GART P22102 15/20 0.55
ATIC P31939 1/20 0.49
CYP1A2 P05177 1/20 0.46
CYP3A4 P08684 1/20 0.46
CYP2C19 P33261 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9038667 0.83 GART (0.64) GARTATIC
SCHEMBL9688062 0.81 GART (0.79) GARTATIC
SCHEMBL9688385 0.80 GART (0.70) GARTATIC
SCHEMBL7607139 0.80 GART (0.49) GART
SCHEMBL10521244 0.80 GART (0.71) GARTATIC
SCHEMBL9794867 0.80 GART (0.66) GARTATIC
SCHEMBL10589282 0.79 GART (0.46) GARTATICCYP1A2CYP3A4CYP2C19
SCHEMBL9794840 0.79 GART (0.66) GARTATIC
SCHEMBL10419882 0.78 GART (0.80) GARTATIC
SCHEMBL9687525 0.78 GART (0.74) GARTATIC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0268377-B1 GLUTAMIC ACID DERIVATIVES, PROCESSES AND INTERMEDIATES FOR THEIR PREPARATION AND PHARMACEUTICAL FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1992-03-18 EP disclosed
US-4940713-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-07-10 US disclosed
US-4880812-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1989-11-14 US disclosed
EP-0268377-A2 Glutamic acid derivatives, processes and intermediates for their preparation and pharmaceutical formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1988-05-25 EP disclosed