SCHEMBL9688929

SCHEMBL9688929

COc1cc2[nH]c(S)nc2c(OC(F)F)c1OC

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATP4A P20648 5/20 0.35
ATP4B P51164 5/20 0.35
GRIN2D O15399 2/20 0.35
GRIN3B O60391 2/20 0.35
GRIN1 Q05586 2/20 0.35
GRIN2A Q12879 2/20 0.35
GRIN2B Q13224 2/20 0.35
GRIN2C Q14957 2/20 0.35
GRIN3A Q8TCU5 2/20 0.35
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
MAOA P21397 2/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
LMNA P02545 2/20 0.33
HPGD P15428 2/20 0.33
CYP2C9 P11712 1/20 0.33
SLC22A2 O15244 1/20 0.33
DDAH1 O94760 1/20 0.33
ABCB1 P08183 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9687854 0.74 MEN1 (0.30) MEN1KMT2A
SCHEMBL9531757 0.74 ATP4A (0.48) ATP4AATP4BGRIN2DGRIN3BGRIN1
SCHEMBL9687316 0.69 NOS2 (0.56) ATP4AATP4BKDM4EALDH1A1LMNA
SCHEMBL9687828 0.69 ATP4A (0.47) ATP4AATP4BKDM4EALDH1A1LMNA
SCHEMBL9686863 0.69 ATP4A (0.41) ATP4AATP4BKDM4EALDH1A1LMNA
SCHEMBL9530579 0.68 ATP4A (0.40) ATP4AATP4BKDM4EATP1A1ATP1B1
SCHEMBL9306374 0.67 CYP3A4 (0.41) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL9793497 0.67 AMY1A (0.35) ATP4AATP4BKDM4EALDH1A1LMNA
SCHEMBL9688009 0.67 ATM (0.37) ATP4AATP4BKDM4EMAPTATP1A1
SCHEMBL2909994 0.66 PDE5A (0.40) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0201575-B1 NEW PICOLINE DERIVATIVES, PREPARATION PROCESS THEREOF, UTILIZATION THEREOF AND DRUGS CONTAINING THEM Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1992-08-12 EP disclosed
US-4686230-A Picoline derivative useful as gastric acid secretion inhibitors BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1987-08-11 US disclosed
EP-0201575-A1 NEW PICOLINE DERIVATIVES, PREPARATION PROCESS THEREOF, UTILIZATION THEREOF AND DRUGS CONTAINING THEM. BYK GULDEN LOMBERG CHEM FAB (DE) 1986-11-20 EP disclosed
WO-1986002646-A1 NEW PICOLINE DERIVATIVES, PREPARATION PROCESS THEREOF, UTILIZATION THEREOF AND DRUGS CONTAINING THEM BYK GULDEN LOMBERG CHEMISCHE FABRIK GESELLSCHAFT M (DE) 1986-05-09 WO disclosed