SCHEMBL9688931

SCHEMBL9688931

Nc1ccc(CCCCCO)c(N)c1N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 3/20 0.37
BCHE P06276 5/20 0.34
ACHE P22303 2/20 0.33
CYP3A4 P08684 2/20 0.33
MAPT P10636 2/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
TLR7 Q9NYK1 1/20 0.31
TYR P14679 2/20 0.31
MEN1 O00255 1/20 0.31
TP53 P04637 1/20 0.31
ALOX5 P09917 1/20 0.31
ALOX15 P16050 1/20 0.31
TSHR P16473 1/20 0.31
HTT P42858 1/20 0.31
KMT2A Q03164 1/20 0.31
TDP1 Q9NUW8 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9687589 0.80 KDM4E (0.40) CA2CYP3A4MAPTKDM4EALDH1A1
SCHEMBL9688930 0.80
SCHEMBL9027471 0.78 TYR (0.43) CYP3A4MAPTKDM4EALDH1A1TYR
SCHEMBL17459905 0.74 RAD52 (0.37) CA2BCHEACHECYP3A4MAPT
SCHEMBL6931597 0.73 CYP3A4 (0.44) CA2BCHECYP3A4MAPTKDM4E
SCHEMBL28124933 0.73 CYP3A4 (0.37) CA2CYP3A4MAPTKDM4EALDH1A1
SCHEMBL19429809 0.73 CYP3A4 (0.44) CA2BCHECYP3A4MAPTKDM4E
SCHEMBL28247926 0.73 LMNA (0.32) MAPTKDM4EMEN1HTTKMT2A
SCHEMBL29154290 0.72 RAD52 (0.38) CA2BCHEACHECYP3A4MAPT
SCHEMBL26944534 0.72 ALDH1A1 (0.41) CA2BCHEACHEALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0511879-A1 Pyrazine derivatives OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1992-11-04 EP disclosed