SCHEMBL9690143

SCHEMBL9690143

CCC(CCC(OS(C)(=O)=O)N1CCNCC1)c1nc(N2CCCC2)nc(N2CCCC2)n1

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 1/20 0.40
USP2 O75604 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
KDM4E B2RXH2 1/20 0.34
HRH4 Q9H3N8 1/20 0.34
HTR2A P28223 3/20 0.34
HTR7 P34969 3/20 0.34
HTR6 P50406 3/20 0.34
CASP1 P29466 1/20 0.33
CASP4 P49662 1/20 0.33
CASP5 P51878 1/20 0.33
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9689052 0.84 CASP1 (0.44) HRH1USP2SMN1; SMN2TDP1HRH4
SCHEMBL9689531 0.78 HRH1 (0.46) HRH1USP2SMN1; SMN2TDP1KDM4E
SCHEMBL9689126 0.72 SLC6A4 (0.37) TDP1KDM4EALDH1A1
SCHEMBL9688175 0.62 CASP1 (0.51) HRH1USP2SMN1; SMN2TDP1HRH4
SCHEMBL8542091 0.62 HRH1 (1.00) HRH1USP2SMN1; SMN2TDP1KDM4E
Hydrochloric Acid SCHEMBL9690244 0.62 CASP1 (0.50) HRH1USP2SMN1; SMN2TDP1HRH4
SCHEMBL778188 0.60 SMN1; SMN2 (1.00) HRH1USP2SMN1; SMN2TDP1KDM4E
SCHEMBL7854614 0.60 SIGMAR1 (0.35)
SCHEMBL3697500 0.58 ALDH1A1 (0.39) KDM4EALDH1A1
SCHEMBL14505381 0.58 HRH1 (0.59) HRH1USP2SMN1; SMN2TDP1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5120843-A Nervous system disorders UPJOHN (US) 1992-06-09 US disclosed
EP-0487510-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1992-05-27 EP disclosed
EP-0358676-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed
EP-0293078-A1 Pharmaceutically active amines THE UPJOHN COMPANY (US) 1988-11-30 EP disclosed
WO-1988008424-A1 PHARMACEUTICALLY ACTIVE AMINES THE UPJOHN COMPANY (US) 1988-11-03 WO disclosed