SCHEMBL9690348

SCHEMBL9690348

N=C(N)NCc1ccc(CCC(=O)O)cc1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 10/20 0.54
FFAR4 Q5NUL3 3/20 0.53
EPHX2 P34913 1/20 0.52
NR1H4 Q96RI1 1/20 0.52
ITGB3 P05106 3/20 0.52
ITGA2B P08514 3/20 0.52
PPARG P37231 1/20 0.51
KEAP1 Q14145 1/20 0.50
CA1 P00915 1/20 0.49
CA2 P00918 1/20 0.49
HTT P42858 1/20 0.46
ST14 Q9Y5Y6 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11788673 0.82 ITGB3 (0.50) FFAR1EPHX2NR1H4ITGB3ITGA2B
SCHEMBL3672272 0.81 CYP2C9 (0.48) CA1CA2ST14
SCHEMBL7303517 0.80 NR1H4 (0.61) FFAR1FFAR4EPHX2NR1H4ITGB3
Trifluoroacetic Acid SCHEMBL28211908 0.80 TMPRSS6 (0.47) FFAR1ITGB3ITGA2BST14
SCHEMBL4109710 0.79 FFAR1 (0.53) FFAR1FFAR4EPHX2NR1H4ITGB3
Hydrochloric Acid SCHEMBL9264373 0.79 NR1H4 (0.60) FFAR1FFAR4EPHX2NR1H4ITGB3
SCHEMBL1916981 0.79 KMT2A (0.62) FFAR1FFAR4EPHX2NR1H4PPARG
SCHEMBL4104833 0.79 KMT2A (0.62) EPHX2NR1H4ST14
Bicarbonate SCHEMBL27358699 0.78 CYP2D6 (0.56) CA1CA2
SCHEMBL27357156 0.78 CA2 (0.45) CA1CA2ST14

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0181592-B1 USE OF SPERGUALIN DERIVATIVES FOR THE PREPARATION OF MEDICAMENTS HAVING IMMUNOSUPPRESSIVE ACTIVITY MICROBIAL CHEMISTRY RESEARCH FOUNDATION (JP) 1992-09-16 EP disclosed
US-4851446-A SPERGUALIN-LIKE GUANIDINES ZAIDAN HOJIN BISEIBUTSU KAGAKU KENKYU KAI (JP) 1989-07-25 US disclosed
EP-0181592-A2 Use of spergualin derivatives for the preparation of medicaments having immunosuppressive activity MICROBIAL CHEMISTRY RESEARCH FOUNDATION (JP) 1986-05-21 EP disclosed