Pyrazine

Pyrazine

SCHEMBL9690748

NC(=O)NC(N)=O.c1cnccn1

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 1/20 0.43
TSHR P16473 3/20 0.37
ADORA3 P0DMS8 2/20 0.37
CYP1A2 P05177 2/20 0.37
CYP3A4 P08684 2/20 0.37
KDM4E B2RXH2 2/20 0.37
MPO P05164 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2A6 P11509 1/20 0.37
CYP2C19 P33261 1/20 0.37
MC4R P32245 1/20 0.37
ADRA1A P35348 1/20 0.37
MC3R P41968 1/20 0.37
NFKB1 P19838 2/20 0.37
CA9 Q16790 2/20 0.37
LMNA P02545 2/20 0.37
MAOA P21397 1/20 0.37
MAOB P27338 1/20 0.37
THPO P40225 1/20 0.37
CA2 P00918 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Pyridine SCHEMBL8567227 0.86 NAPRT (0.47) CRBNTSHRADORA3CYP1A2CYP3A4
Pyrazine SCHEMBL27913358 0.81 CYP1A2 (0.62) TSHRADORA3CYP1A2CYP3A4KDM4E
Pyrazine SCHEMBL28327835 0.79 ALDH1A1 (0.50) TSHRADORA3CYP1A2CYP3A4KDM4E
SCHEMBL15045 0.79
SCHEMBL27939070 0.79 CRBN (0.60) CRBNTSHRCYP1A2CYP3A4KDM4E
SCHEMBL27524722 0.79 CRBN (0.60) CRBNTSHRCYP1A2CYP3A4KDM4E
SCHEMBL27560286 0.79 CRBN (0.60) CRBNTSHRCYP1A2CYP3A4KDM4E
Pyrazine SCHEMBL4712089 0.76 ACHE (0.54) TSHRADORA3CYP1A2CYP3A4KDM4E
Pyrazine SCHEMBL306074 0.76 ACHE (0.54) TSHRADORA3CYP1A2CYP3A4KDM4E
Benzene SCHEMBL27729594 0.76 CRBN (0.50) CRBNTSHRCYP1A2CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0229391-B1 PIPERIDINE DERIVATE, ITS USE AND PHARMACEUTICAL COMPOSITION CONTAINING IT Eisai Co., Ltd. (JP) 1992-07-29 EP claimed
CN-110317321-A Quinoid conjugated polymer and preparation method and application thereof 东莞理工学院 2019-10-11 CN disclosed