SCHEMBL9045462

SCHEMBL9045462

CC1=C(OC(=O)OC(C)C)C(c2ccc(Cl)c(Cl)c2)C2=C(COC2=O)N1C

nearest known ligand 0.38

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 9/20 0.38
TSHR P16473 1/20 0.34
PYGL P06737 1/20 0.32
PYGM P11217 1/20 0.32
SLC6A4 P31645 8/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
MAPT P10636 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HTT P42858 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
ADORA2B P29275 1/20 0.32
LMNA P02545 1/20 0.32
ABCC9 O60706 1/20 0.31
KCNJ11 Q14654 1/20 0.31
SLC6A2 P23975 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8080875 0.86 ADORA2B (0.41) SLC6A3TSHRPYGLPYGMNPSR1
SCHEMBL9829012 0.79 KDM4E (0.33) TSHRCYP1A2CYP3A4MAPTCYP2C9
SCHEMBL9690849 0.77 KDM4E (0.39) NPSR1LMNA
SCHEMBL9829022 0.73 PYGL (0.48) PYGLPYGM
SCHEMBL9828158 0.71 PYGM (0.35) PYGLPYGM
SCHEMBL10653759 0.70 CYP3A4 (0.39) SLC6A3TSHRPYGLPYGMCYP3A4
SCHEMBL9045340 0.70 PYGL (0.36) SLC6A3TSHRPYGLPYGMCYP1A2
SCHEMBL9827653 0.70 PYGM (0.35) PYGLPYGM
SCHEMBL10968852 0.69 PYGM (0.37) TSHRPYGLPYGM
SCHEMBL8441182 0.69 NPSR1 (0.44) SLC6A3TSHRSLC6A4NPSR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0705830-A1 2,3-Cyclic condensed 1,4-dihydropyridines, process for their preparation and their use as K-channel modulators BAYER AG (DE) 1996-04-10 EP disclosed