SCHEMBL9690993

SCHEMBL9690993

c1cnc(NCCN2CCC(Nc3nc4cccnc4n3Cc3cccs3)C2)nc1

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SLC6A9 P48067 1/20 0.46
MAPT P10636 8/20 0.38
ENPP2 Q13822 1/20 0.37
EED O75530 1/20 0.37
TP53 P04637 4/20 0.36
ROCK2 O75116 1/20 0.36
CCR2 P41597 1/20 0.36
ROCK1 Q13464 1/20 0.36
POLB P06746 1/20 0.35
CXCR4 P61073 1/20 0.35
SSTR5 P35346 1/20 0.35
KCNH2 Q12809 1/20 0.35
PYGM P11217 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Fumaric Acid SCHEMBL9630608 0.93 SLC6A9 (0.43) SLC6A9MAPTENPP2TP53POLB
SCHEMBL9629312 0.89 SLC6A9 (0.47) SLC6A9MAPTENPP2EEDTP53
SCHEMBL9690741 0.87 SLC6A9 (0.46) SLC6A9MAPTENPP2TP53POLB
SCHEMBL9691136 0.87 SLC6A9 (0.44) SLC6A9MAPTENPP2EEDTP53
SCHEMBL9690941 0.85 HRH1 (0.41) MAPTEEDTP53ROCK2ROCK1
SCHEMBL9629649 0.84 SLC6A9 (0.44) SLC6A9MAPTENPP2EEDTP53
Fumaric Acid SCHEMBL9630404 0.84 SLC6A9 (0.43) SLC6A9MAPTENPP2TP53POLB
SCHEMBL9629371 0.84 HTR1A (0.42) SLC6A9MAPTEEDTP53CXCR4
SCHEMBL10753371 0.83 SLC6A9 (0.49) SLC6A9MAPTENPP2TP53POLB
SCHEMBL9538015 0.81 SLC6A9 (0.65) SLC6A9MAPTENPP2TP53POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0297661-B1 [(Bicyclic heterocyclyl)methyl and -hetero] substituted hexahydro-1H-azepines and pyrrolidines JANSSEN PHARMACEUTICA N.V. (BE) 1992-09-16 EP disclosed