SCHEMBL9691809

SCHEMBL9691809

COC(=O)OC1=C(C)NC2=C(C(=O)OC3(CCCCC3)C2)C1c1ccccc1[N+](=O)[O-]

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 6/20 0.46
MAPT P10636 5/20 0.46
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 4/20 0.46
ADORA3 P0DMS8 3/20 0.46
LMNA P02545 3/20 0.46
TDP1 Q9NUW8 3/20 0.46
ABCC4 O15439 2/20 0.46
CACNA1F O60840 2/20 0.46
ABCB11 O95342 2/20 0.46
CYP1A2 P05177 2/20 0.46
ADORA2A P29274 2/20 0.46
ADORA1 P30542 2/20 0.46
OPRM1 P35372 2/20 0.46
SCN1A P35498 2/20 0.46
HTR2B P41595 2/20 0.46
CACNA1D Q01668 2/20 0.46
KCNH2 Q12809 2/20 0.46
CACNA1S Q13698 2/20 0.46
CACNA1C Q13936 2/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11009533 0.87 MAPT (0.60) KMT2AMAPTALDH1A1KDM4EADORA3
SCHEMBL11111322 0.83 ALDH1A1 (0.51) KMT2AMAPTALDH1A1KDM4EADORA3
SCHEMBL6427770 0.78 ADORA3 (0.67) KMT2AMAPTALDH1A1KDM4EADORA3
SCHEMBL10369519 0.76 ADORA3 (0.58) KMT2AMAPTALDH1A1KDM4EADORA3
SCHEMBL11116098 0.76 KMT2A (0.44) KMT2AMAPTALDH1A1KDM4EADORA3
SCHEMBL9838777 0.75 ALDH1A1 (0.52) KMT2AMAPTALDH1A1KDM4EADORA3
SCHEMBL9689499 0.75 ADORA3 (0.62) KMT2AMAPTALDH1A1KDM4EADORA3
SCHEMBL11360822 0.75 ADORA3 (0.62) KMT2AMAPTALDH1A1KDM4EADORA3
SCHEMBL11114191 0.74 CACNA1C (0.53) KMT2AMAPTALDH1A1KDM4EADORA3
SCHEMBL6425245 0.74 CACNA1D (0.61) KMT2AMAPTALDH1A1KDM4EADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed
EP-0071819-B1 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1987-04-22 EP disclosed