SCHEMBL9691902

SCHEMBL9691902

CCOC(=O)OC1=C(C)NC(C)=C(OC(=O)O)C1c1ccccc1OCc1cccc([N+](=O)[O-])c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE1C Q14123 1/20 0.49
ADORA3 P0DMS8 2/20 0.47
MEN1 O00255 5/20 0.46
KMT2A Q03164 5/20 0.46
ALDH1A1 P00352 2/20 0.46
CACNA1F O60840 8/20 0.46
CACNA1D Q01668 8/20 0.46
CACNA1S Q13698 8/20 0.46
CACNA1C Q13936 8/20 0.46
HIF1A Q16665 3/20 0.45
MAPT P10636 3/20 0.45
CYP1A2 P05177 2/20 0.45
CYP3A4 P08684 2/20 0.45
CYP2C9 P11712 2/20 0.45
CYP2C19 P33261 2/20 0.45
POLB P06746 2/20 0.45
LMNA P02545 1/20 0.45
MAPK1 P28482 1/20 0.45
GPR55 Q9Y2T6 1/20 0.45
CYP2D6 P10635 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9690786 0.94 MEN1 (0.48) PDE1CADORA3MEN1KMT2AALDH1A1
SCHEMBL9691516 0.84 ADORA3 (0.44) PDE1CADORA3MEN1KMT2AALDH1A1
SCHEMBL11004215 0.82 PDE1C (0.56) PDE1CADORA3MEN1KMT2AALDH1A1
SCHEMBL11004220 0.82 PDE1C (0.56) PDE1CADORA3MEN1KMT2AALDH1A1
SCHEMBL9691692 0.82 KMT2A (0.43) MEN1KMT2AALDH1A1MAPTPOLB
SCHEMBL9691359 0.81 POLB (0.44) MEN1KMT2AALDH1A1MAPTPOLB
SCHEMBL10817795 0.81 ABCB1 (0.46) MAPT
SCHEMBL11371616 0.80 CACNA1F (0.66) PDE1CADORA3MEN1KMT2ACACNA1F
SCHEMBL9691807 0.80 SLC1A5 (0.44) MAPTFFAR1
SCHEMBL9691796 0.80 HTR6 (0.43) LMNAFFAR1SIRT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed
EP-0071819-B1 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1987-04-22 EP disclosed