SCHEMBL9691807

SCHEMBL9691807

COC(=O)OC1=C(C)NC(C)=C(OC(=O)O)C1c1ccccc1OCc1cccc(OC)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
SLC1A5 Q15758 1/20 0.44
MTNR1A P48039 3/20 0.43
MTNR1B P49286 2/20 0.43
ABCB1 P08183 4/20 0.42
HTR1A P08908 3/20 0.42
DRD2 P14416 2/20 0.42
AKR1C3 P42330 1/20 0.41
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
LRRK2 Q5S007 1/20 0.40
KDM4E B2RXH2 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
FFAR1 O14842 1/20 0.40
MRGPRX4 Q96LA9 2/20 0.40
MMP13 P45452 1/20 0.40
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10817795 0.95 ABCB1 (0.46) SLC1A5MTNR1AMTNR1BABCB1HTR1A
SCHEMBL9691359 0.90 POLB (0.44) HTR1AKDM4EMAPTHTTSMN1; SMN2
SCHEMBL9691796 0.89 HTR6 (0.43) AKR1C3KDM4EFFAR1MRGPRX4
SCHEMBL10914095 0.87 POLB (0.46) HTR1AKDM4EMAPTHTTSMN1; SMN2
SCHEMBL9690850 0.87 GAA (0.40) KDM4EFFAR1MAPTHTTSMN1; SMN2
SCHEMBL9690786 0.86 MEN1 (0.48) ABCB1HTR1AADRA1DADRA1AADRA1B
SCHEMBL9689534 0.86 FFAR4 (0.44) SLC1A5MRGPRX4
SCHEMBL9691648 0.85 TP53 (0.41) SLC1A5KDM4EMAPTHTTSMN1; SMN2
SCHEMBL9690877 0.85 HTR6 (0.43) HTR1AKDM4EFFAR1MAPT
SCHEMBL9691625 0.85 NR1I2 (0.42) SLC1A5HTR1AKDM4EMAPTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0071819-B2 DIHYDROPYRIDINES WITH A POSITIVE INOTROPIC ACTIVITY, THEIR USE IN PHARMACEUTICAL PREPARATIONS, AND PROCESSES FOR THEIR PREPARATION BAYER AG (DE) 1992-06-10 EP disclosed