SCHEMBL9694041

SCHEMBL9694041

O=[N+]([O-])c1cccc(F)c1C(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 4/20 0.47
GPR35 Q9HC97 2/20 0.45
HSPB1 P04792 1/20 0.41
ALDH1A1 P00352 3/20 0.41
TSHR P16473 3/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ATM Q13315 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
HIF1A Q16665 2/20 0.40
S100A4 P26447 1/20 0.40
MAPT P10636 2/20 0.40
MAPK1 P28482 2/20 0.40
POLB P06746 1/20 0.40
HSD17B10 Q99714 1/20 0.39
AR P10275 1/20 0.39
CYP3A4 P08684 1/20 0.39
HPGD P15428 1/20 0.39
ALOX15 P16050 1/20 0.39
TXNRD1 Q16881 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11521456 0.85 ATM (0.49) TDP1HSPB1ALDH1A1TSHRMEN1
SCHEMBL29044667 0.84 TDP1 (0.47) TDP1GPR35HSPB1ALDH1A1MEN1
SCHEMBL17109851 0.83 TDP1 (0.48) TDP1GPR35HSPB1ALDH1A1TSHR
SCHEMBL1995565 0.81 TDP1 (0.47) TDP1GPR35ALDH1A1TSHRMEN1
SCHEMBL16953540 0.79 TDP1 (0.45) TDP1GPR35ALDH1A1TSHRMEN1
SCHEMBL4728834 0.79 HPGD (0.46) TDP1GPR35ALDH1A1TSHRMEN1
SCHEMBL10338398 0.79 TSHR (0.58) TDP1GPR35ALDH1A1TSHRMEN1
SCHEMBL9905068 0.79 TDP1 (0.45) TDP1GPR35ALDH1A1TSHRSMN1; SMN2
SCHEMBL11375306 0.79 GPR35 (0.56) TDP1GPR35ALDH1A1TSHRSMN1; SMN2
SCHEMBL4520380 0.79 TDP1 (0.45) TDP1GPR35ALDH1A1TSHRMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110088086-A Disubstituted maleic amide class connexon and its preparation method and application for antibody-drug conjugate 迈威(上海)生物科技有限公司 2019-08-02 CN disclosed
CN-109810039-A Disubstituted maleimide-based linker for antibody-drug coupling, preparation method and application thereof 上海青润医药科技有限公司 2019-05-28 CN disclosed
CN-106458939-B * oxazolidinyl compound and the selective androgen receptor agonist comprising the compound 东亚ST株式会社 2019-05-17 CN disclosed
CN-109071563-A Inhibitors of bruton's tyrosine kinase and methods of use thereof 詹森药业有限公司 2018-12-21 CN disclosed
CN-108431001-A Ring-fused pyrimidines compound or its salt 大鹏药品工业株式会社 2018-08-21 CN disclosed
CN-104884453-B Anthelmintic compounds and compositions and methods of using the same 梅里亚股份有限公司 2018-06-22 CN disclosed
CN-105339355-B Novel CYP17 inhibitor/antiandrogen 奥赖恩公司 2018-02-27 CN disclosed
CN-107652293-A Imidazopyridazines IRAK4 inhibitor and its preparation method and application 中国药科大学 2018-02-02 CN disclosed
CN-106029661-B Pyrazolo [1,5-A ] pyridine derivatives and methods of use thereof 亚尼塔公司 2017-11-03 CN disclosed
CN-107257793-A Anti- worm compound, composition and its application method 梅里亚股份有限公司 2017-10-17 CN disclosed
CN-101821266-B Modulators of cystic fibrosis transmembrane channel regulators VERTEX PHARMA 2014-03-12 CN disclosed
CN-102459186-A Anthelmintic agents and uses thereof ANTHELMINTIC AGENTS AND THEIR USE 2012-05-16 CN disclosed
CN-1863789-A Substituted isoquinolinones PORTOLA PHARM INC (US) 2006-11-15 CN disclosed
EP-0270964-B1 PROCESS FOR OBTAINING SUBSTITUTED FLUOROBENZENES BAYER AG (DE) 1992-07-08 EP disclosed
US-4868347-A SOLVENT EXTRACTION BAYER AKTIENGESELLSCHAFT (DE) 1989-09-19 US disclosed
EP-0270964-A2 Process for obtaining substituted fluorobenzenes BAYER AG (DE) 1988-06-15 EP disclosed
US-4224340-A Anti-inflammatory compositions containing α-phenyl-N-phenylnitrone compounds WILLIAM H. RORER, INC. (US) 1980-09-23 US disclosed
US-4214003-A ANTIINFLAMMATORY AGENTS WILLIAM H. RORER, INC. (US) 1980-07-22 US disclosed
US-4197314-A WITH A DIPHENYL NITRONE WILLIAM H. RORER, INC. (US) 1980-04-08 US disclosed
US-4153722-A ANTIINFLAMMATORY, A-PHENYL-N-PHENYLNITRONE WILLIAM H. RORER, INC. (US) 1979-05-08 US disclosed