SCHEMBL9905068

SCHEMBL9905068

O=[N+]([O-])c1cccc(I)c1C(F)(F)F

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 3/20 0.45
GPR35 Q9HC97 2/20 0.44
ALDH1A1 P00352 4/20 0.40
TSHR P16473 3/20 0.40
P2RY6 Q15077 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
S100A4 P26447 1/20 0.39
AR P10275 1/20 0.38
HSD17B10 Q99714 1/20 0.38
CYP3A4 P08684 1/20 0.38
HPGD P15428 1/20 0.38
ALOX15 P16050 1/20 0.38
HIF1A Q16665 1/20 0.38
TXNRD1 Q16881 1/20 0.38
TXNRD3 Q86VQ6 1/20 0.38
TXNRD2 Q9NNW7 1/20 0.38
P2RX1 P51575 2/20 0.37
POLB P06746 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1995565 0.79 TDP1 (0.47) TDP1GPR35ALDH1A1TSHRSMN1; SMN2
SCHEMBL9694041 0.79 TDP1 (0.47) TDP1GPR35ALDH1A1TSHRSMN1; SMN2
SCHEMBL4520380 0.78 TDP1 (0.45) TDP1GPR35ALDH1A1TSHRSMN1; SMN2
SCHEMBL28303063 0.78 ALDH1A1 (0.46) TDP1GPR35ALDH1A1TSHRSMN1; SMN2
SCHEMBL10338398 0.78 TSHR (0.58) TDP1GPR35ALDH1A1TSHRSMN1; SMN2
SCHEMBL4728834 0.78 HPGD (0.46) TDP1GPR35ALDH1A1TSHRP2RY6
SCHEMBL16953540 0.78 TDP1 (0.45) TDP1GPR35ALDH1A1TSHRSMN1; SMN2
SCHEMBL11375306 0.78 GPR35 (0.56) TDP1GPR35ALDH1A1TSHRSMN1; SMN2
SCHEMBL27733344 0.76 ALDH1A1 (0.45) TDP1GPR35ALDH1A1TSHRHSD17B10
SCHEMBL10768517 0.75 ERN1 (0.57) TDP1GPR35ALDH1A1TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011072241-A9 4-OXO-1H-QUINOLINE-3-CARBOXAMIDES AS MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-06-14 WO disclosed