SCHEMBL9694976

SCHEMBL9694976

CCOC(=O)CSc1cc(N=C=O)c(F)cc1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.39
TSHR P16473 3/20 0.39
HSD17B10 Q99714 3/20 0.39
CYP1A2 P05177 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
ALOX15 P16050 1/20 0.39
CYP2C19 P33261 1/20 0.39
KDM4E B2RXH2 4/20 0.36
HPGD P15428 3/20 0.36
TP53 P04637 1/20 0.36
HTT P42858 1/20 0.36
MAPT P10636 2/20 0.36
LMNA P02545 3/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
TYMS P04818 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8604172 0.89 ALDH1A1 (0.39) ALDH1A1TSHRHSD17B10CYP1A2CYP3A4
SCHEMBL8484111 0.88 ALDH1A1 (0.42) ALDH1A1TSHRHSD17B10CYP1A2CYP3A4
SCHEMBL8603927 0.81 ALDH1A1 (0.38) ALDH1A1TSHRHSD17B10CYP1A2CYP3A4
SCHEMBL9569006 0.80 MAPT (0.37) ALDH1A1HSD17B10CYP1A2CYP3A4CYP2C9
SCHEMBL8601643 0.80 ALDH1A1 (0.40) ALDH1A1TSHRHSD17B10CYP1A2CYP3A4
SCHEMBL8603065 0.79 KDM4E (0.48) ALDH1A1TSHRHSD17B10CYP1A2CYP3A4
SCHEMBL8600331 0.78 ALDH1A1 (0.39) ALDH1A1TSHRHSD17B10CYP1A2CYP3A4
SCHEMBL8485382 0.77 ALDH1A1 (0.41) ALDH1A1TSHRHSD17B10CYP1A2CYP3A4
SCHEMBL10916815 0.76 CYP4F2 (0.47) TSHRCYP1A2CYP2C19HPGDMAPT
SCHEMBL9851167 0.76 BCL2L11 (0.41) ALDH1A1TSHRHSD17B10CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0484776-A1 Arylsubstituted alkyliden-nitrogenheterocycles BAYER AG (DE) 1992-05-13 EP disclosed
EP-0416361-A1 N-(5-alkyl thiophenyl)-nitrogenheterocycles BAYER AG (DE) 1991-03-13 EP disclosed