SCHEMBL9695041

SCHEMBL9695041

CC(C)c1c(CO)c(-c2ccc(F)cc2)c2n1CCCC2

nearest known ligand 0.42

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GCGR P47871 13/20 0.42
THRB P10828 1/20 0.39
TGFBR1 P36897 1/20 0.39
PTGS2 P35354 2/20 0.38
KMT2A Q03164 1/20 0.37
PTGS1 P23219 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9780839 0.82 ALDH1A1 (0.34) GCGRTHRBTGFBR1PTGS2KMT2A
SCHEMBL9696143 0.79 KMT2A (0.53) PTGS2KMT2APTGS1
SCHEMBL9695099 0.79 PTGS2 (0.39) PTGS2KMT2APTGS1
SCHEMBL9696155 0.77 KMT2A (0.35) GCGRTHRBTGFBR1PTGS2KMT2A
SCHEMBL9697138 0.76 KMT2A (0.34) GCGRTHRBTGFBR1PTGS2KMT2A
SCHEMBL9696224 0.73 HMGCR (0.38) THRB
SCHEMBL9696237 0.73 HMGCR (0.37) THRB
SCHEMBL9696231 0.73 HMGCR (0.37) THRB
SCHEMBL6290810 0.71 RIPK3 (0.45) KMT2A
SCHEMBL2654771 0.69 GCGR (0.67) GCGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5124453-A Treatment of corresponding aldehyde with lithium bis(tri-methylsilyl)amide E. R. SQUIBB & SONS, INC. (US) 1992-06-23 US disclosed
EP-0444532-A1 Phosphorus-containing HMG-CoA reductase inhibitors, new intermediates and method E.R. SQUIBB & SONS, INC. (US) 1991-09-04 EP disclosed
US-5025000-A Anticholesterol, antilipemic agents E. R. SQUIBB & SONS, INC. (US) 1991-06-18 US disclosed