SCHEMBL9696155

SCHEMBL9696155

CC(C)c1c(C=C(Cl)Cl)c(-c2ccc(F)cc2)c2n1CCCC2

nearest known ligand 0.35

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.35
GCGR P47871 3/20 0.34
PTGS2 P35354 2/20 0.34
PTGS1 P23219 1/20 0.34
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KCNK3 O14649 2/20 0.32
THRB P10828 2/20 0.31
TGFBR1 P36897 2/20 0.31
ALOX5 P09917 2/20 0.31
HTR1A P08908 2/20 0.31
DRD2 P14416 2/20 0.31
HTR2A P28223 2/20 0.31
HTR7 P34969 2/20 0.31
HTR6 P50406 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9695099 0.85 PTGS2 (0.39) KMT2APTGS2PTGS1ALDH1A1KCNK3
SCHEMBL9696229 0.79 KMT2A (0.43) KMT2AGCGRPTGS2PTGS1KDM4E
SCHEMBL9695041 0.77 GCGR (0.42) KMT2AGCGRPTGS2PTGS1THRB
SCHEMBL9696143 0.76 KMT2A (0.53) KMT2APTGS2PTGS1KDM4EALDH1A1
SCHEMBL9697138 0.76 KMT2A (0.34) KMT2AGCGRPTGS2PTGS1KDM4E
SCHEMBL9780839 0.72 ALDH1A1 (0.34) KMT2AGCGRPTGS2PTGS1ALDH1A1
SCHEMBL9696399 0.65 KMT2A (0.45) KMT2APTGS2PTGS1KDM4EALDH1A1
SCHEMBL9696167 0.63 KMT2A (0.43) KMT2AKDM4EALDH1A1TDP1KCNK3
SCHEMBL9697147 0.62 KMT2A (0.67) KMT2AKDM4EALDH1A1TDP1KCNK3
SCHEMBL6486123 0.60 PTGES (0.49) KMT2APTGS2PTGS1THRBTGFBR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5124453-A Treatment of corresponding aldehyde with lithium bis(tri-methylsilyl)amide E. R. SQUIBB & SONS, INC. (US) 1992-06-23 US disclosed
EP-0444532-A1 Phosphorus-containing HMG-CoA reductase inhibitors, new intermediates and method E.R. SQUIBB & SONS, INC. (US) 1991-09-04 EP disclosed
US-5025000-A Anticholesterol, antilipemic agents E. R. SQUIBB & SONS, INC. (US) 1991-06-18 US disclosed