SCHEMBL9699330

SCHEMBL9699330

O=NN1c2ccccc2OCC1CN1CCCCC1

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.53
ADRA2B P18089 1/20 0.53
ADRA2C P18825 1/20 0.53
ADRA1D P25100 1/20 0.53
ADRA1A P35348 1/20 0.53
ADRA1B P35368 1/20 0.53
SCN1A P35498 1/20 0.53
SCN2A Q99250 1/20 0.53
SCN3A Q9NY46 1/20 0.53
LTA4H P09960 4/20 0.41
ABCB1 P08183 2/20 0.39
ALDH1A1 P00352 2/20 0.39
DRD2 P14416 1/20 0.38
HTR1A P08908 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
LMNA P02545 1/20 0.38
HPGD P15428 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9699366 0.88 GAA (0.48) LTA4HALDH1A1
SCHEMBL9700614 0.80 ADRA2A (0.57) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9699310 0.80 NOTUM (0.38) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9701406 0.79 SMN1; SMN2 (0.37) ADRA2AADRA1AALDH1A1HTR1ALMNA
SCHEMBL9699297 0.77 NOTUM (0.38) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9699253 0.76 ADRA2A (0.42) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9699236 0.74 LTA4H (0.40) LTA4HALDH1A1LMNAHPGDSMN1; SMN2
SCHEMBL9701674 0.73 ADRA2A (0.42) ADRA2AADRA2BADRA2CADRA1DADRA1A
Piperoxan SCHEMBL12503311 0.72 ADRA2A (0.97) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9700406 0.71 ADRB1 (0.38) ADRA2CDRD2HTR1ASIGMAR1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed