SCHEMBL9699366

SCHEMBL9699366

O=NN1c2ccccc2OCC1CN1CCOCC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GAA P10253 2/20 0.48
CNR1 P21554 4/20 0.43
CNR2 P34972 4/20 0.43
ALDH1A1 P00352 3/20 0.43
MAPT P10636 1/20 0.43
NPC1 O15118 1/20 0.43
MTOR P42345 1/20 0.43
RAB9A P51151 1/20 0.43
LTA4H P09960 3/20 0.43
CYP3A4 P08684 2/20 0.42
MEN1 O00255 1/20 0.42
CYP2C9 P11712 1/20 0.42
KMT2A Q03164 1/20 0.42
CYP2D6 P10635 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9699330 0.88 ADRA2A (0.53) ALDH1A1LTA4H
SCHEMBL9700311 0.80 GAA (0.51) GAACNR1CNR2ALDH1A1MAPT
SCHEMBL25434899 0.80 GAA (0.51) GAACNR1CNR2ALDH1A1MAPT
SCHEMBL9701406 0.78 SMN1; SMN2 (0.37) GAAALDH1A1MAPTNPC1RAB9A
SCHEMBL9699315 0.78 CNR1 (0.47) GAACNR1CNR2ALDH1A1MAPT
SCHEMBL9699236 0.73 LTA4H (0.40) GAAALDH1A1NPC1RAB9ALTA4H
SCHEMBL9700502 0.71 ADRA2A (0.45) GAALTA4HKMT2A
SCHEMBL9699297 0.71 NOTUM (0.38) ALDH1A1
SCHEMBL9699310 0.71 NOTUM (0.38) ALDH1A1
SCHEMBL9701449 0.68 DRD2 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed