SCHEMBL9700522

SCHEMBL9700522

c1ccc2c(c1)NCC(CC1CNCCCN1)O2

nearest known ligand 0.40

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 2/20 0.39
CASR P41180 1/20 0.39
HTR1A P08908 3/20 0.38
HPGD P15428 1/20 0.36
LTA4H P09960 1/20 0.33
CXCR4 P61073 1/20 0.32
POLB P06746 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701381 0.76 LTA4H (0.33) LTA4HCXCR4
SCHEMBL9699300 0.73 SLC6A2 (0.32) CXCR4
SCHEMBL4824743 0.71 HPGD (0.51) NISCHCASRHTR1AHPGDPOLB
SCHEMBL30112409 0.70 CASR (0.50) NISCHCASRHTR1AHPGDPOLB
SCHEMBL8570483 0.70 CASR (0.47) NISCHCASRHTR1AHPGD
SCHEMBL3969657 0.70 CASR (0.47) NISCHCASRHTR1AHPGD
SCHEMBL17150937 0.70 CASR (0.50) NISCHCASRHTR1AHPGDPOLB
SCHEMBL3969660 0.70 CASR (0.47) NISCHCASRHTR1AHPGD
SCHEMBL2638179 0.70 CASR (0.47) NISCHCASRHTR1AHPGD
SCHEMBL9700525 0.70 HTR1A (0.47) NISCHCASRHTR1ACXCR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed