SCHEMBL9700865

SCHEMBL9700865

Cc1nc(C)n(-c2cccc3c2NC(=O)OC3)c1C

nearest known ligand 0.33

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
TYMS P04818 1/20 0.33
CYP1A2 P05177 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
HSD17B10 Q99714 1/20 0.33
GRM5 P41594 1/20 0.32
GAA P10253 1/20 0.32
MB P02144 1/20 0.32
HCAR1 Q9BXC0 3/20 0.31
CYP11B1 P15538 2/20 0.30
CYP11B2 P19099 2/20 0.30
POLB P06746 1/20 0.30
PTPN11 Q06124 1/20 0.30
MAOA P21397 1/20 0.30
MAOB P27338 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL436140 0.72 HTR5A (0.44) KDM4EALDH1A1TYMSCYP1A2HPGD
SCHEMBL3605239 0.66 MAOA (0.37) KDM4EALDH1A1TYMSCYP1A2HPGD
SCHEMBL3605242 0.66 MAOA (0.37) KDM4EALDH1A1TYMSCYP1A2HPGD
SCHEMBL14805480 0.66 ALDH1A1 (0.39) KDM4EALDH1A1TYMSCYP1A2HPGD
SCHEMBL24711772 0.62 HTR1A (0.33) KDM4EALDH1A1TYMSCYP1A2HPGD
SCHEMBL12030669 0.61 GAA (0.59) KDM4EALDH1A1GAAPOLB
SCHEMBL464780 0.58 AHR (0.50) KDM4EALDH1A1TYMSCYP1A2HPGD
SCHEMBL20881863 0.58 MAPT (0.47) KDM4EALDH1A1CYP1A2CYP2C19HSD17B10
SCHEMBL9700774 0.57 ALDH1A1 (0.32) ALDH1A1
SCHEMBL10959840 0.57 AHR (0.45) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0510235-A1 Novel benzoxazine or benzothiazine derivatives and process for the preparation of the same DONG-A PHARM. CO., LTD. (KR) 1992-10-28 EP disclosed