SCHEMBL9701377

SCHEMBL9701377

CC(=O)CC(=O)c1cccc2cccnc12

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.58
NPC1 O15118 3/20 0.54
RAB9A P51151 3/20 0.54
CASP3 P42574 1/20 0.54
SENP8 Q96LD8 1/20 0.54
SENP7 Q9BQF6 1/20 0.54
SENP6 Q9GZR1 1/20 0.54
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
ALDH1A1 P00352 4/20 0.50
KDR P35968 2/20 0.50
TDP1 Q9NUW8 2/20 0.48
POLB P06746 2/20 0.48
LMNA P02545 1/20 0.48
ALOX12 P18054 1/20 0.48
MAPT P10636 2/20 0.47
HPGD P15428 1/20 0.47
HSD17B10 Q99714 1/20 0.47
KDM4E B2RXH2 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12883029 0.83 PARP1 (0.62) PARP1NPC1RAB9ACASP3SENP8
SCHEMBL30144797 0.81 PARP1 (0.68) PARP1NPC1RAB9ACASP3SENP8
SCHEMBL2632726 0.81 PARP1 (0.68) PARP1NPC1RAB9ACASP3SENP8
Phenanthroline SCHEMBL7693062 0.81 TDP1 (0.61) PARP1ALDH1A1TDP1POLBLMNA
SCHEMBL3886554 0.80 PARP1 (0.62) PARP1NPC1RAB9ACASP3SENP8
SCHEMBL15228399 0.80 PARP1 (0.62) PARP1NPC1RAB9ACASP3SENP8
SCHEMBL16581134 0.80 PARP1 (0.62) PARP1NPC1RAB9ACASP3SENP8
Phenanthroline SCHEMBL27590762 0.80 TDP1 (0.59) PARP1ALDH1A1TDP1POLBLMNA
Oxyquinoline SCHEMBL27460253 0.79 MMP2 (0.70) PARP1RAB9AMEN1KMT2AALDH1A1
SCHEMBL11808999 0.78 P2RX7 (0.62) NPC1RAB9AMEN1KMT2AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed