SCHEMBL9701379

SCHEMBL9701379

COc1ccc2ccc(C(=O)CC(C)=O)cc2c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.61
ALDH1A1 P00352 3/20 0.61
HPGD P15428 2/20 0.61
HSD17B10 Q99714 2/20 0.61
CYP2C19 P33261 1/20 0.61
KDM4E B2RXH2 4/20 0.58
NPC1 O15118 4/20 0.51
RAB9A P51151 4/20 0.51
SMN1; SMN2 Q16637 3/20 0.51
LMNA P02545 2/20 0.51
TP53 P04637 1/20 0.51
CYP3A4 P08684 1/20 0.51
MAPT P10636 1/20 0.51
MAOA P21397 1/20 0.51
SLC6A2 P23975 1/20 0.51
SLC6A3 Q01959 1/20 0.51
PLAU P00749 1/20 0.50
PKM P14618 1/20 0.48
CASP3 P42574 1/20 0.48
SENP7 Q9BQF6 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11247310 0.97 ALDH1A1 (0.65) CYP1A2ALDH1A1HPGDHSD17B10CYP2C19
SCHEMBL2603411 0.82 CYP1A2 (0.67) CYP1A2ALDH1A1HPGDHSD17B10CYP2C19
SCHEMBL2774094 0.82 SMN1; SMN2 (0.72) CYP1A2ALDH1A1HPGDHSD17B10CYP2C19
SCHEMBL1374066 0.81 ALDH1A1 (0.64) ALDH1A1HSD17B10NPC1RAB9ALMNA
SCHEMBL31427513 0.80 ALDH1A1 (0.69) CYP1A2ALDH1A1HPGDHSD17B10CYP2C19
SCHEMBL7173547 0.80 ALDH1A1 (0.69) CYP1A2ALDH1A1HPGDHSD17B10CYP2C19
SCHEMBL545959 0.80 KDM4E (0.66) CYP1A2ALDH1A1HPGDHSD17B10CYP2C19
SCHEMBL29242089 0.80 NPC1 (0.60) ALDH1A1HPGDHSD17B10KDM4ENPC1
SCHEMBL12532275 0.79 NPC1 (0.64) CYP1A2ALDH1A1HPGDHSD17B10CYP2C19
SCHEMBL2644205 0.79 ALDH1A1 (0.58) CYP1A2ALDH1A1HPGDHSD17B10CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed