SCHEMBL9701474

SCHEMBL9701474

CCCOc1ccc(-c2ccc(-c3nnn[nH]3)c(=O)[nH]2)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 4/20 0.41
CYP2C9 P11712 4/20 0.41
CYP3A4 P08684 3/20 0.41
CYP2D6 P10635 3/20 0.41
CYP19A1 P11511 3/20 0.41
CYP2C19 P33261 3/20 0.41
RAB9A P51151 6/20 0.41
NPC1 O15118 5/20 0.41
TP53 P04637 3/20 0.41
HSD17B10 Q99714 3/20 0.41
GAA P10253 1/20 0.41
GPR84 Q9NQS5 1/20 0.40
MAPT P10636 3/20 0.39
SMN1; SMN2 Q16637 5/20 0.39
HPGD P15428 3/20 0.39
ALDH1A1 P00352 2/20 0.39
ALOX12 P18054 1/20 0.39
CTSV O60911 1/20 0.37
CTSL P07711 1/20 0.37
KDM4E B2RXH2 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701387 0.95 CYP2C9 (0.47) CYP1A2CYP2C9CYP3A4CYP2D6CYP19A1
SCHEMBL9700689 0.90 RAB9A (0.33) CYP1A2RAB9ANPC1TP53HSD17B10
SCHEMBL9526113 0.87 MAPT (0.41) CYP1A2CYP2C9CYP3A4CYP2D6CYP19A1
SCHEMBL9701582 0.85 GCGR (0.39) CYP1A2CYP2C9HSD17B10MAPTSMN1; SMN2
SCHEMBL9700644 0.84 PDE5A (0.38) CYP1A2RAB9ANPC1HSD17B10GAA
SCHEMBL9525805 0.84 CDC7 (0.36) CYP2C9GAAMAPTALOX12KDM4E
SCHEMBL9701382 0.84 SMN1; SMN2 (0.42) CYP1A2CYP2C9CYP2D6CYP19A1CYP2C19
SCHEMBL9524898 0.83 PDE4A (0.37) NPC1HSD17B10MAPTHPGDALDH1A1
SCHEMBL7644729 0.81 PDE5A (0.47) CYP1A2HSD17B10MAPTSMN1; SMN2HPGD
SCHEMBL9701433 0.80 PDE5A (0.33) CYP1A2MAPTHPGDALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992006085-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-04-16 WO claimed
WO-1992006085-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-04-16 WO disclosed