SCHEMBL9701602

SCHEMBL9701602

NN1c2cccc(Cl)c2OCC1CN1CCCC1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.38
ADRA2B P18089 1/20 0.38
ADRA2C P18825 1/20 0.38
ADRA1D P25100 1/20 0.38
ADRA1A P35348 1/20 0.38
ADRA1B P35368 1/20 0.38
SCN1A P35498 1/20 0.38
SCN2A Q99250 1/20 0.38
SCN3A Q9NY46 1/20 0.38
NOTUM Q6P988 1/20 0.36
KDM4E B2RXH2 1/20 0.35
ALDH1A1 P00352 1/20 0.35
POLB P06746 1/20 0.35
SIGMAR1 Q99720 2/20 0.33
HRH3 Q9Y5N1 1/20 0.33
DRD2 P14416 3/20 0.33
DRD4 P21917 3/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
OPRK1 P41145 1/20 0.32
CHRNA7 P36544 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9699278 0.97 NOTUM (0.36) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9699323 0.90 CXCR4 (0.36) ADRA2CSIGMAR1HRH3DRD2
SCHEMBL9699340 0.89 CYP2A13 (0.39) NOTUMDRD2DRD4
SCHEMBL9728710 0.89 DRD2 (0.40) NOTUMHRH3DRD2DRD4LTA4H
SCHEMBL9699310 0.82 NOTUM (0.38) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9699269 0.82 NOTUM (0.38) NOTUMDRD2SMN1; SMN2
SCHEMBL9700351 0.81 ADRA2A (0.41) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9699297 0.80 NOTUM (0.38) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9701613 0.79 ADRA2A (0.41) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL9700368 0.77 NOTUM (0.37) ADRA1DADRA1AADRA1BNOTUM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed