SCHEMBL9701613

SCHEMBL9701613

COc1cccc2c1OCC(CN1CCC1)N2N

nearest known ligand 0.41

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
ADRA2C P18825 1/20 0.41
ADRA1A P35348 10/20 0.39
HTR1A P08908 9/20 0.39
ADRA1D P25100 8/20 0.39
ADRA1B P35368 7/20 0.39
POLB P06746 2/20 0.36
DRD2 P14416 2/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
OPRM1 P35372 1/20 0.36
OPRD1 P41143 1/20 0.36
OPRK1 P41145 1/20 0.36
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700351 0.98 ADRA2A (0.41) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL9699337 0.91 ADRA2A (0.42) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL9699287 0.90 HTR7 (0.40) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL9728617 0.90 ADRA1A (0.41) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL9700158 0.83 HTR2A (0.38) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL10378979 0.83 ADRA1A (0.38) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL9701674 0.82 ADRA2A (0.42) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL9699278 0.81 NOTUM (0.36) ADRA2AADRA2BADRA2CADRA1AADRA1D
SCHEMBL9699253 0.80 ADRA2A (0.42) ADRA2AADRA2BADRA2CADRA1AHTR1A
SCHEMBL9700327 0.80 ADRA1D (0.38) ADRA2AADRA2BADRA2CADRA1AHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed