SCHEMBL9701642

SCHEMBL9701642

COc1ccccc1N1CCN(CCC2CCc3onc(-c4cccc(F)c4)c3C2=O)C(I)C1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 6/20 0.43
DRD2 P14416 6/20 0.39
HTR2A P28223 2/20 0.39
TACR3 P29371 1/20 0.39
KDM4E B2RXH2 1/20 0.36
ALDH1A1 P00352 1/20 0.36
GAA P10253 1/20 0.36
DRD4 P21917 4/20 0.36
DRD3 P35462 4/20 0.36
MAPT P10636 2/20 0.36
THRB P10828 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36
ADRA1B P35368 1/20 0.36
MEN1 O00255 1/20 0.36
GFER P55789 1/20 0.36
KMT2A Q03164 1/20 0.36
HTR7 P34969 1/20 0.36
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700487 0.88 HTR2C (0.43) HTR2CDRD2HTR2AKDM4EALDH1A1
SCHEMBL9024747 0.88 HTR2C (0.57) HTR2CDRD2HTR2ATACR3DRD4
SCHEMBL9024113 0.77 HTR2C (0.54) HTR2CDRD2ALDH1A1DRD4DRD3
SCHEMBL9687660 0.76 HTR2C (0.56) HTR2CDRD2HTR2ADRD4DRD3
Hydrochloric Acid SCHEMBL9023938 0.75 HTR2C (0.56) HTR2CDRD2HTR2ADRD4DRD3
SCHEMBL9474916 0.72 HTR2C (0.53) HTR2CDRD2DRD4MAPTADRA1D
SCHEMBL9688546 0.72 HTR2C (0.56) HTR2CDRD2HTR2AKDM4EALDH1A1
SCHEMBL9445139 0.72 HDAC1 (0.41) HTR2CDRD2HTR2AHTR7
Hydrochloric Acid SCHEMBL9445171 0.71 HTR2C (0.53) HTR2CDRD2DRD4MAPTADRA1D
Hydrochloric Acid SCHEMBL9023951 0.71 HTR2C (0.55) HTR2CDRD2HTR2AKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0474012-A1 6,7-Dihydro-3-phenyl-1,2-benzisoxazol-4(5H)-ones and -ols, a process for their preparation and their use as medicaments HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-03-11 EP disclosed