SCHEMBL9701693

SCHEMBL9701693

COc1cc2c3c(c1)cc(C)n3C(CN1CCSCC1)CO2

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.35
KDM4E B2RXH2 2/20 0.35
CNR1 P21554 4/20 0.33
CNR2 P34972 4/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
ADRA2A P08913 1/20 0.31
ADRA2B P18089 1/20 0.31
ADRA2C P18825 1/20 0.31
MAPT P10636 1/20 0.30
NPC1 O15118 1/20 0.30
MTOR P42345 1/20 0.30
RAB9A P51151 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9701569 0.90 CNR1 (0.34) ALDH1A1CNR1CNR2MEN1KMT2A
SCHEMBL9700053 0.90 CNR1 (0.34) CNR1CNR2MEN1KMT2ACYP3A4
SCHEMBL9700282 0.88 HRH3 (0.41) KDM4ECNR1CNR2MEN1KMT2A
SCHEMBL9728633 0.84 L3MBTL1 (0.36) ALDH1A1CNR1CNR2MEN1KMT2A
SCHEMBL9699311 0.83 ADRB1 (0.32) CNR1CNR2MEN1KMT2ACYP3A4
SCHEMBL9701634 0.81 DRD2 (0.30)
SCHEMBL9701364 0.74 CNR1 (0.38) ALDH1A1KDM4ECNR1CNR2MEN1
SCHEMBL9701369 0.74 CNR1 (0.51) ALDH1A1CNR1CNR2MEN1KMT2A
SCHEMBL9699289 0.73 CNR1 (0.33) ALDH1A1CNR1CNR2MEN1KMT2A
SCHEMBL9701537 0.73 HRH3 (0.34) ALDH1A1CNR1CNR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5112820-A Vision defects STERLING DRUG INC. (US) 1992-05-12 US disclosed
US-5109135-A 2- or 3-aminomethyl-4-amino-3,4-dihydro-2H-1,4-benzoxazine intermediates STERLING DRUG INC. (US) 1992-04-28 US disclosed
US-5066803-A Chemical intermediates for analgesics STERLING DRUG INC. (US) 1991-11-19 US disclosed
WO-1990007505-A1 2- AND 3-AMINOMETHYL-6-ARYLCARBONYL-2,3-DIHYDROPYRROLO[1,2,3-de]-1,4-BENZOXAZINES STERLING DRUG INC. (US) 1990-07-12 WO disclosed
US-4939138-A 2- and 3-aminomethyl-6-arylcarbonyl-2,3-dihydropyrrolo(1,2,3-DE)-1,4-benzoxazines STERLING DRUG INC. (US) 1990-07-03 US disclosed