SCHEMBL9702587

SCHEMBL9702587

CCCCSc1ccccc1-c1ccc(-c2nnn[nH]2)c(=O)[nH]1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.41
HTT P42858 2/20 0.41
KDM4E B2RXH2 2/20 0.41
TSHR P16473 1/20 0.41
SMN1; SMN2 Q16637 4/20 0.38
MAPT P10636 4/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
GAA P10253 1/20 0.38
PDE5A O76074 2/20 0.37
PTGS2 P35354 4/20 0.35
S100A4 P26447 1/20 0.35
SOAT1 P35610 1/20 0.35
HPGD P15428 1/20 0.34
POLB P06746 2/20 0.33
LMNA P02545 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
XDH P47989 1/20 0.33
CTSB P07858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9700772 0.80 XDH (0.35) ALDH1A1HTTKDM4ETSHRSMN1; SMN2
SCHEMBL9588370 0.76 KDM4E (0.40) ALDH1A1HTTKDM4ETSHRSMN1; SMN2
SCHEMBL7644729 0.76 PDE5A (0.47) ALDH1A1KDM4ESMN1; SMN2MAPTMEN1
SCHEMBL9525926 0.76 CYP2C9 (0.31) ALDH1A1HTTKDM4ETSHRMAPT
SCHEMBL9530230 0.74 MDM2 (0.41) ALDH1A1HTTKDM4ETSHRSMN1; SMN2
SCHEMBL9702603 0.72
SCHEMBL9701387 0.72 CYP2C9 (0.47) SMN1; SMN2HPGDPOLBLMNAXDH
SCHEMBL9535284 0.72 KDM4E (0.41) KDM4EGAAPOLB
SCHEMBL9701382 0.70 SMN1; SMN2 (0.42) ALDH1A1KDM4ETSHRSMN1; SMN2MAPT
SCHEMBL9700783 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992006085-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-04-16 WO claimed
WO-1992006085-A1 PHENYLPYRIDINOL DERIVATIVES AS MEDICAMENTS SMITH KLINE & FRENCH LABORATORIES LIMITED (GB) 1992-04-16 WO disclosed