SCHEMBL9703250

SCHEMBL9703250

Oc1ccc2[nH]cc(C3CCC(CCN4CCN(c5ccccn5)CC4)CC3)c2c1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 5/20 0.79
DRD3 P35462 4/20 0.79
DRD4 P21917 2/20 0.79
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
THPO P40225 1/20 0.50
USP2 O75604 1/20 0.46
ALDH1A1 P00352 1/20 0.46
MAPK1 P28482 1/20 0.46
HSD17B10 Q99714 1/20 0.46
HTR1A P08908 1/20 0.46
HTR2A P28223 1/20 0.46
HTR2C P28335 1/20 0.46
HTR7 P34969 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9703912 0.89 DRD2 (0.79) DRD2DRD3DRD4HTR1AHTR2A
SCHEMBL9703331 0.89 DRD2 (1.00) DRD2DRD3DRD4
SCHEMBL9703684 0.87 DRD2 (0.75) DRD2DRD3DRD4HTR1A
SCHEMBL9703158 0.79 DRD2 (0.81) DRD2DRD3DRD4HTR1A
SCHEMBL9703330 0.79 DRD2 (0.81) DRD2DRD3DRD4CYP2D6
SCHEMBL19823060 0.75 DRD2 (0.66) DRD2DRD3DRD4HTR1AHTR2A
SCHEMBL9703913 0.73 DRD2 (0.66) DRD2DRD3DRD4HTR1AHTR2A
SCHEMBL9703731 0.73 DRD2 (0.68) DRD2DRD3DRD4CYP1A2CYP3A4
SCHEMBL9773160 0.72 DRD2 (0.70) DRD2DRD3DRD4HTR1AHTR2A
SCHEMBL3849926 0.72 DRD2 (0.70) DRD2DRD3DRD4HTR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992012977-A1 SUBSTITUTED INDOLES AS CENTRAL NERVOUS SYSTEM AGENTS WARNER-LAMBERT COMPANY (US) 1992-08-06 WO claimed
WO-1992012977-A1 SUBSTITUTED INDOLES AS CENTRAL NERVOUS SYSTEM AGENTS WARNER-LAMBERT COMPANY (US) 1992-08-06 WO disclosed
US-5124332-A Dopaminergic agents, hypotensive agents WARNER-LAMBERT COMPANY (US) 1992-06-23 US disclosed