SCHEMBL9703372

SCHEMBL9703372

COc1cc(SC)ccc1-c1nc2cc3c(cc2[nH]1)CC(C)(C)C(=O)N3

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
AMY1A P0DUB6 11/20 0.38
PDE3B Q13370 2/20 0.36
PDE3A Q14432 2/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
PDE5A O76074 1/20 0.36
CHEK2 O96017 1/20 0.36
NPC1 O15118 1/20 0.34
HSP90AA1 P07900 1/20 0.34
PKM P14618 1/20 0.34
RAB9A P51151 1/20 0.34
MAPK1 P28482 1/20 0.34
AURKA O14965 1/20 0.33
AURKB Q96GD4 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9703536 0.87 TP53 (0.42) AMY1APDE3BPDE3APDE4APDE4B
SCHEMBL9703453 0.84 AMY1A (0.37) AMY1APDE3BPDE3APDE4APDE4B
SCHEMBL10373868 0.81 PDE3B (0.49) AMY1APDE3BPDE3APDE4APDE4B
SCHEMBL10697003 0.78 AMY1A (0.45) AMY1APDE3BPDE3APDE4APDE4B
SCHEMBL10557582 0.77 AMY1A (0.39) AMY1APDE3BPDE3APDE5ACHEK2
SCHEMBL9703298 0.77 PDE5A (0.38) AMY1APDE3BPDE3APDE4APDE4B
SCHEMBL9703397 0.77 NPC1 (0.50) PDE3BPDE3APDE4APDE4BPDE4C
SCHEMBL10849719 0.76 AMY1A (0.41) AMY1APDE3BPDE3APDE5ACHEK2
SCHEMBL11301435 0.74 AMY1A (0.38) AMY1APDE3BPDE3APDE5ACHEK2
SCHEMBL9703459 0.73 PDE4A (0.50) PDE3BPDE3APDE4APDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5116843-A Anticoagulants, hypotensive agents and cardiovascular disorder BOEHRINGER MANNHEIM GMBH (DE) 1992-05-26 US disclosed
EP-0275888-A2 Tricyclic benzimidazoles, process for their preparation and use as medicaments Roche Diagnostics GmbH (DE) 1988-07-27 EP disclosed