SCHEMBL9703975

SCHEMBL9703975

CCCCc1nc2nc(Br)ccc2[nH]1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.40
PI4KA P42356 1/20 0.39
PI4K2B Q8TCG2 1/20 0.39
PI4K2A Q9BTU6 1/20 0.39
PI4KB Q9UBF8 1/20 0.39
NOS3 P29474 2/20 0.39
NOS1 P29475 2/20 0.39
NOS2 P35228 2/20 0.39
ALDH1A1 P00352 1/20 0.38
MAPK1 P28482 1/20 0.38
GSK3B P49841 1/20 0.38
POLB P06746 1/20 0.38
KMT2A Q03164 1/20 0.37
GPR84 Q9NQS5 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9318008 0.83 DDAH1 (0.46) NOS3NOS1NOS2
SCHEMBL10439327 0.81 PARP1 (0.40) PARP1PI4KAPI4K2BPI4K2API4KB
SCHEMBL9704776 0.81 PI4KA (0.46) PARP1PI4KAPI4K2BPI4K2API4KB
SCHEMBL8641790 0.79 PARP1 (0.39) PARP1PI4KAPI4K2BPI4K2API4KB
SCHEMBL9705920 0.78 PRMT5 (0.41) PARP1PI4KAPI4K2BPI4K2API4KB
SCHEMBL31586691 0.75 SMN1; SMN2 (0.39) NOS3NOS1NOS2ALDH1A1MAPK1
SCHEMBL7853172 0.75 HPGD (0.46) PI4KAPI4K2BPI4K2API4KBNOS3
SCHEMBL8326986 0.74 NOS1 (0.54) NOS3NOS1NOS2POLB
SCHEMBL9704371 0.72 SMN1; SMN2 (0.48) ALDH1A1MAPK1
SCHEMBL7850823 0.72 NOS3 (0.38) PI4KAPI4K2BPI4K2API4KBNOS3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0470543-A1 Heterocyclic imidazoles, remedies containing them and processes for their preparation Dr. Karl Thomae GmbH (DE) 1992-02-12 EP disclosed