SCHEMBL9704

SCHEMBL9704

Clc1ncnc2sccc12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 1/20 0.59
AURKA O14965 1/20 0.59
DAPK3 O43293 1/20 0.59
JAK2 O60674 1/20 0.59
MAP4K4 O95819 1/20 0.59
ABL1 P00519 1/20 0.59
NTRK1 P04629 1/20 0.59
LCK P06239 1/20 0.59
FYN P06241 1/20 0.59
CSF1R P07333 1/20 0.59
RET P07949 1/20 0.59
IGF1R P08069 1/20 0.59
MET P08581 1/20 0.59
PDGFRB P09619 1/20 0.59
PIM1 P11309 1/20 0.59
FGFR1 P11362 1/20 0.59
PRKACA P17612 1/20 0.59
LTK P29376 1/20 0.59
KDR P35968 1/20 0.59
MAP2K2 P36507 1/20 0.59

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7255700 0.89 CHEK1 (0.49) CHEK1AURKADAPK3JAK2MAP4K4
SCHEMBL2843606 0.76 CHEK1 (0.61) CHEK1AURKADAPK3JAK2MAP4K4
SCHEMBL1192489 0.74 CHEK1 (0.59) CHEK1AURKADAPK3JAK2MAP4K4
SCHEMBL8018832 0.74 CHEK1 (0.59) CHEK1AURKADAPK3JAK2MAP4K4
SCHEMBL22412847 0.74 CHEK1 (0.59) CHEK1AURKADAPK3JAK2MAP4K4
SCHEMBL968490 0.74 DYRK1A (1.00) CHEK1AURKADAPK3JAK2MAP4K4
SCHEMBL30958678 0.74 CHEK1 (0.59) CHEK1AURKADAPK3JAK2MAP4K4
SCHEMBL12559905 0.74 CHEK1 (0.59) CHEK1AURKADAPK3JAK2MAP4K4
SCHEMBL29365779 0.74 DYRK1A (1.00) CHEK1AURKADAPK3JAK2MAP4K4
SCHEMBL2919086 0.71 DYRK1A (0.45) CHEK1AURKADAPK3JAK2MAP4K4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 384 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118146226-A Pyrrolo [2,3-d ] pyrimidine compound with nitrogen-containing heterocyclic structure, and preparation method and application thereof 贵州大学 2024-06-07 CN claimed
CN-122036605-A Antagonists of GPR39 proteins 俄勒冈健康科学大学 2026-05-15 CN disclosed
US-20260132147-A1 BAX INHIBITORS AND USES THEREOF CASE WESTERN RESERVE UNIV (US) 2026-05-14 US disclosed
US-12479857-B2 Bax inhibitors and uses thereof CASE WESTERN RESERVE UNIVERSITY (US) 2025-11-25 US disclosed
US-20250282785-A1 PYRROLIDINONE DERIVATIVES AS INHIBITORS OF NF KAPPA B INDUCING KINASE JANSSEN PHARMACEUTICA NV (BE) 2025-09-11 US disclosed
US-12390463-B2 Dosage forms and regimens for amino acid compounds PLIANT THERAPEUTICS, INC. (US) 2025-08-19 US disclosed
US-20250223288-A1 AMINO ACID COMPOUNDS AND METHODS OF USE PLIANT THERAPEUTICS, INC. 2025-07-10 US disclosed
EP-4522608-A1 PYRROLIDINONE DERIVATIVES AS INHIBITORS OF NF KAPPA B INDUCING KINASE JANSSEN Pharmaceutica NV (BE) 2025-03-19 EP disclosed
EP-4520329-A2 TREATMENT OF RESPIRATORY DISEASES WITH AMINO ACID COMPOUNDS Pliant Therapeutics, Inc. (US) 2025-03-12 EP disclosed
EP-4509512-A2 AMINO ACID COMPOUNDS AND METHODS OF USE Pliant Therapeutics, Inc. (US) 2025-02-19 EP disclosed
EP-0370704-A2 Aralkylamine derivatives, preparation thereof and fungicides containing the same UBE INDUSTRIES, LTD. (JP) 1990-05-30 EP disclosed
EP-0196524-B1 PHENOXYALKYLAMINOPYRIMIDINE DERIVATIVES, THEIR PREPARATION AND INSECTICIDAL AND ACARICIDAL COMPOSITIONS CONTAINING THEM SANKYO COMPANY LIMITED (JP) 1990-03-07 EP disclosed
US-4845097-A AGRICULTURE SANKYO COMPANY LIMITED (JP) 1989-07-04 US disclosed
EP-0103114-B1 THIENOPYRIDINE DERIVATIVES, THEIR PREPARATION AND INSECTICIDAL AND ACARICIDAL COMPOSITIONS CONTAINING THEM SANKYO COMPANY LIMITED (JP) 1986-11-12 EP disclosed
EP-0196524-A2 Phenoxyalkylaminopyrimidine derivatives, their preparation and insecticidal and acaricidal compositions containing them SANKYO COMPANY LIMITED (JP) 1986-10-08 EP disclosed
US-4562193-A 4-[2-(Di- or trisubstitutedphenoxy)ethyl amino]thienodipyrimidines and insecticidal and acaricidal composition containing said pyrimidines SANKYO COMPANY LIMITED (JP) 1985-12-31 US disclosed
EP-0103114-A2 Thienopyridine derivatives, their preparation and insecticidal and acaricidal compositions containing them SANKYO COMPANY LIMITED (JP) 1984-03-21 EP disclosed
US-4256738-A BACTERICIDES, PYRIMIDINYL, QUINAZOLINYL BOEHRINGER INGELHEIM GMBH (DE) 1981-03-17 US disclosed
US-4196207-A Process for controlling eradicating or preventing infestations of animals by Ixodid ticks ICI AUSTRALIA LIMITED 1980-04-01 US disclosed
US-4146716-A PLANT GROWTH REGULATORS, FUNGICIDES, BACTERICIDES, VIRICIDES, INSECTICIDES IMPERIAL CHEMICAL INDUSTRIES LIMITED (GB) 1979-03-27 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260132147-A1 BAX INHIBITORS AND USES THEREOF BAX, BCL2, BAK1 CHEK1 326/4885AURKA 3878/4885DAPK3 108/4885
US-12390463-B2 Dosage forms and regimens for amino acid compounds ITGB6, ITGA6, ITGAV CHEK1 3817/4885AURKA 3839/4885DAPK3 3807/4885
US-20250223288-A1 AMINO ACID COMPOUNDS AND METHODS OF USE ITGB6, ITGA6, ITGA5 CHEK1 3709/4885AURKA 3420/4885DAPK3 2805/4885
US-20250282785-A1 PYRROLIDINONE DERIVATIVES AS INHIBITORS OF NF KAPPA B INDUCING KINASE NFKBIA, IKBKG, IKBKB CHEK1 1018/4885AURKA 3029/4885DAPK3 49/4885
US-12479857-B2 Bax inhibitors and uses thereof BAX, TMBIM6, BCL2 CHEK1 299/4885AURKA 2706/4885DAPK3 98/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.