SCHEMBL9704225

SCHEMBL9704225

COc1cc2ccnc(-c3ccccc3F)c2cc1OC

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 2/20 0.51
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
CYP3A4 P08684 3/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
ACHE P22303 2/20 0.48
MAOA P21397 1/20 0.44
PDE10A Q9Y233 3/20 0.44
USP2 O75604 2/20 0.44
ALDH1A1 P00352 2/20 0.44
LMNA P02545 2/20 0.44
MAPK1 P28482 2/20 0.44
PDE3B Q13370 2/20 0.44
PDE3A Q14432 2/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
HIF1A Q16665 2/20 0.44
RAB9A P51151 2/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9704512 0.84 TRPA1 (0.52) TRPA1MEN1KMT2ACYP3A4CYP1A2
SCHEMBL10333393 0.81 KLK7 (0.50) TRPA1MEN1KMT2ACYP3A4CYP1A2
SCHEMBL10333713 0.79 MEN1 (0.46) TRPA1MEN1KMT2ACYP3A4CYP1A2
Bromide SCHEMBL8002743 0.78 MEN1 (0.60) MEN1KMT2ACYP3A4CYP1A2CYP2D6
SCHEMBL15674510 0.75 MAP4K1 (0.45) CYP3A4CYP1A2CYP2D6CYP2C19PDE10A
SCHEMBL28068055 0.74 MAOA (0.47) MEN1KMT2AACHEMAOATNF
SCHEMBL18257430 0.74 APEX1 (0.43) LMNASMN1; SMN2MAPT
SCHEMBL4655563 0.73 MEN1 (0.55) TRPA1MEN1KMT2ACYP3A4CYP1A2
SCHEMBL2460475 0.73 MEN1 (0.66) TRPA1MEN1KMT2ACYP3A4CYP1A2
SCHEMBL14341090 0.72 CYP1A2 (0.47) TRPA1MEN1KMT2ACYP3A4CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-1992011242-A1 FUNGICIDAL ISOQUINOLINE DERIVATIVES SHELL INTERNATIONALE RESEARCH MAATSCHAPPIJ B.V. (NL) 1992-07-09 WO disclosed
EP-0491441-A1 Fungicidal isoquinoline derivatives SHELL INTERNATIONALE RESEARCHMAATSCHAPPIJ B.V. (NL) 1992-06-24 EP disclosed