SCHEMBL10333393

SCHEMBL10333393

COc1cc2ccnc(-c3ccccc3SC)c2cc1OC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KLK7 P49862 2/20 0.50
KLK14 Q9P0G3 2/20 0.50
KLK5 Q9Y337 2/20 0.50
CTSG P08311 1/20 0.50
CTRC Q99895 1/20 0.50
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
ACHE P22303 2/20 0.46
TNF P01375 2/20 0.44
MAOA P21397 1/20 0.43
CYP3A4 P08684 3/20 0.42
PDE10A Q9Y233 3/20 0.42
USP2 O75604 2/20 0.42
ALDH1A1 P00352 2/20 0.42
LMNA P02545 2/20 0.42
CYP1A2 P05177 2/20 0.42
CYP2D6 P10635 2/20 0.42
CYP2C9 P11712 2/20 0.42
MAPK1 P28482 2/20 0.42
CYP2C19 P33261 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9704225 0.81 TRPA1 (0.51) MEN1KMT2AACHETNFMAOA
SCHEMBL10334046 0.78 MEN1 (0.44) MEN1KMT2AACHECYP3A4ALDH1A1
SCHEMBL10333713 0.76 MEN1 (0.46) MEN1KMT2AACHETNFMAOA
Bromide SCHEMBL8002743 0.76 MEN1 (0.60) MEN1KMT2AACHECYP3A4PDE10A
SCHEMBL28068055 0.72 MAOA (0.47) MEN1KMT2AACHETNFMAOA
SCHEMBL2460475 0.71 MEN1 (0.66) MEN1KMT2AACHETNFCYP3A4
SCHEMBL9704512 0.70 TRPA1 (0.52) MEN1KMT2AACHETNFCYP3A4
Hydrochloric Acid SCHEMBL1022954 0.70 MEN1 (0.64) MEN1KMT2AACHETNFCYP3A4
SCHEMBL954159 0.69 ALDH1A1 (0.54) MEN1KMT2AMAOACYP3A4PDE10A
SCHEMBL30789068 0.69 MEN1 (0.59) MEN1KMT2AACHETNFCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4900751-A 2-Pyridinyl-phenyl-sulphinyl-and-phenyl-thio-benzimidazoles having antiflammatory or gastic acid secretion inhibition activity FISONS PLC (GB) 1990-02-13 US disclosed
EP-0283504-A1 COMPOUNDS FISONS plc (GB) 1988-09-28 EP disclosed
WO-1988002367-A1 COMPOUNDS FISONS PLC (GB) 1988-04-07 WO disclosed
EP-0262845-A1 Heterocyclic substituted azole derivatives FISONS plc (GB) 1988-04-06 EP disclosed