SCHEMBL9704526

SCHEMBL9704526

CCN1c2ncccc2NC(=O)c2c1nc(C)c(Cl)c2C

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.37
CHRM2 P08172 4/20 0.35
LMNA P02545 2/20 0.35
CHRM1 P11229 2/20 0.35
USP2 O75604 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CHRM4 P08173 1/20 0.35
CHRM5 P08912 1/20 0.35
CYP2D6 P10635 1/20 0.35
CHRM3 P20309 1/20 0.35
GMNN O75496 1/20 0.34
APEX1 P27695 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8303480 0.79 CYP3A4 (0.40) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL9704205 0.78 LMNA (0.42) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL9703875 0.77 CYP2C9 (0.42) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL8300334 0.75 RAB9A (0.50) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL9704536 0.74 RAB9A (0.42) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL9705868 0.71 CYP2C9 (0.45) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL9369774 0.69 RAB9A (0.59) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL8888719 0.68 ALDH1A1 (0.45) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL4031265 0.68 RAB9A (0.43) RAB9ACHRM2LMNACHRM1USP2
SCHEMBL9704218 0.66 CYP2C9 (0.47) RAB9ACHRM2LMNAALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0482481-A1 Method for the preparation of 5,11-dihydro-6H-dipyrido[3,2-b:2',3'-e][1,4]diazepines BOEHRINGER INGELHEIM PHARMACEUTICALS INC. (US) 1992-04-29 EP disclosed