SCHEMBL9705360

SCHEMBL9705360

N#CN1Cc2ccccc2-c2ccccc2C1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSL P07711 1/20 0.47
CTSB P07858 1/20 0.47
CTSK P43235 1/20 0.47
USP7 Q93009 6/20 0.46
KMT2A Q03164 1/20 0.43
TEAD1 P28347 3/20 0.43
TEAD4 Q15561 3/20 0.43
TEAD2 Q15562 3/20 0.43
ADRA1D P25100 1/20 0.42
ADRA1A P35348 1/20 0.42
ADRA1B P35368 1/20 0.42
IDO1 P14902 1/20 0.41
SMN1; SMN2 Q16637 3/20 0.38
NPC1 O15118 2/20 0.38
RAB9A P51151 2/20 0.38
LMNA P02545 2/20 0.38
TEAD3 Q99594 1/20 0.37
KDM4E B2RXH2 3/20 0.36
HSD17B10 Q99714 2/20 0.36
HPGD P15428 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22061852 0.88 CTSL (0.52) CTSLCTSBCTSKUSP7KMT2A
SCHEMBL19357687 0.78 UCHL1 (0.49) CTSLCTSBCTSKUSP7TEAD1
SCHEMBL19357728 0.77 TEAD1 (0.47) CTSLCTSBCTSKUSP7TEAD1
SCHEMBL29710088 0.77 TEAD1 (0.47) CTSLCTSBCTSKUSP7TEAD1
SCHEMBL19357626 0.75 TEAD1 (0.46) CTSLCTSBCTSKUSP7TEAD1
SCHEMBL2327219 0.74 MAOA (0.52) CTSLCTSBCTSKUSP7KMT2A
SCHEMBL30043742 0.74 MAOA (0.52) CTSLCTSBCTSKUSP7KMT2A
SCHEMBL19375056 0.72 TEAD1 (0.43) CTSLCTSBCTSKUSP7KMT2A
SCHEMBL20608442 0.71 UCHL1 (0.46) USP7TEAD1TEAD4TEAD2TEAD3
SCHEMBL13939593 0.69 KMT2A (0.48) KMT2AADRA1DADRA1AADRA1BIDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0192034-B1 DIBENZAZEPINE DERIVATIVES, THEIR PREPARATION, STARTING MATERIALS FOR THEIR PREPARATION, AND USE OF THE DIBENZAZEPINE DERIVATIVES AS PESTICIDES CIBA-GEIGY AG (CH) 1992-07-15 EP claimed
US-4833245-A CHEMICAL INTERMEDIATES FOR INSECTICIDES HOFFMANN-LA ROCHE INC. (US) 1989-05-23 US claimed
EP-0192034-A2 Dibenzazepine derivatives, their preparation, starting materials for their preparation, and use of the dibenzazepine derivatives as pesticides CIBA-GEIGY AG (CH) 1986-08-27 EP claimed
EP-0192034-B1 DIBENZAZEPINE DERIVATIVES, THEIR PREPARATION, STARTING MATERIALS FOR THEIR PREPARATION, AND USE OF THE DIBENZAZEPINE DERIVATIVES AS PESTICIDES CIBA-GEIGY AG (CH) 1992-07-15 EP disclosed
US-5015640-A Insecticides or miticides CIBA-GEIGY CORPORATION (US) 1991-05-14 US disclosed
EP-0368176-A1 Esters of carboximidic acid, their preparation, and their use as pesticides CIBA-GEIGY AG (CH) 1990-05-16 EP disclosed
US-4833245-A CHEMICAL INTERMEDIATES FOR INSECTICIDES HOFFMANN-LA ROCHE INC. (US) 1989-05-23 US disclosed
US-4766115-A 5,6-dihydro-6H-dibenz[c,e]azepine-6-(thio)carboximidic acid esters and insecticidal use thereof HOFFMANN-LA ROCHE INC. (US) 1988-08-23 US disclosed
EP-0192034-A2 Dibenzazepine derivatives, their preparation, starting materials for their preparation, and use of the dibenzazepine derivatives as pesticides CIBA-GEIGY AG (CH) 1986-08-27 EP disclosed