SCHEMBL9705668

SCHEMBL9705668

Cc1cc(CCCCCOc2c(Cl)cc(C#N)cc2C(F)(F)F)on1

nearest known ligand 0.45

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.45
CYP3A4 P08684 1/20 0.45
CYP2D6 P10635 1/20 0.45
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
LRRK2 Q5S007 1/20 0.30
CYP11B1 P15538 1/20 0.30
CYP11B2 P19099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9211432 0.89 NR1I2 (0.41) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL8875626 0.85 NR1I2 (0.45) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL9863089 0.81 MRGPRX4 (0.42) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL9705898 0.81 NR1I2 (0.46) NR1I2CYP3A4CYP2D6
SCHEMBL9208044 0.80 NR1I2 (0.50) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL9876491 0.78 ICMT (0.44) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL9705747 0.77 NR1I2 (0.43) NR1I2CYP3A4CYP2D6
SCHEMBL8136926 0.77 NR1I2 (0.45) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL9862969 0.76 ICMT (0.44) NR1I2CYP3A4CYP2D6MEN1KMT2A
SCHEMBL8134990 0.76 NR1I2 (0.47) NR1I2CYP3A4CYP2D6MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0207454-B1 ISOXAZOLE AND FURAN DERIVATIVES, THEIR PREPARATION AND USE AS ANTIVIRAL AGENTS STERLING WINTHROP INC. (US) 1992-09-09 EP disclosed
US-5002960-A Viricides for combating picornaviruses STERLING DRUG, INC. (US) 1991-03-26 US disclosed
US-4939267-A Viricides STERLING DRUG INC. (US) 1990-07-03 US disclosed
US-4843087-A OXAZOLINYL COMPOUNDS; RHINOVIRUSES AND PICORNAVIRUSES STERLING DRUG INC. (US) 1989-06-27 US disclosed
EP-0207454-A2 Isoxazole and furan derivatives, their preparation and use as antiviral agents STERLING WINTHROP INC. (US) 1987-01-07 EP disclosed